SCHEMBL21948720

SCHEMBL21948720

CC(C)c1cnc2n(N)cccc1-2

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 1/20 0.33
FEN1 P39748 1/20 0.33
DHFR P00374 1/20 0.31
P2RX3 P56373 1/20 0.31
P2RX2 Q9UBL9 1/20 0.31
CA1 P00915 2/20 0.31
CA2 P00918 2/20 0.31
CA12 O43570 1/20 0.31
CA9 Q16790 1/20 0.31
TRPA1 O75762 1/20 0.30
FAAH O00519 1/20 0.30
LMNA P02545 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
GABRA1 P14867 1/20 0.30
HPGD P15428 1/20 0.30
TSHR P16473 1/20 0.30
GABRB1 P18505 1/20 0.30
GABRG2 P18507 1/20 0.30
PTGS1 P23219 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12914173 0.81 MC4R (0.30) ALOX5APFEN1CA1CA2TRPA1
SCHEMBL21964686 0.70 USP1 (0.33)
SCHEMBL21764022 0.68 FAAH (0.40) CA1CA2CA12CA9FAAH
SCHEMBL23132917 0.67 NR1I2 (0.33) CA1CA2FAAHLMNACYP1A2
SCHEMBL18438723 0.66
SCHEMBL18729638 0.63 CYP1A2 (0.46) ALOX5APFEN1LMNACYP1A2CYP3A4
SCHEMBL13863865 0.63 BRD4 (0.51) TSHRHTR2CPIP4K2C
SCHEMBL23879670 0.63 CYP1A2 (0.46) ALOX5APFEN1LMNACYP1A2CYP3A4
SCHEMBL2737326 0.63 NR1I2 (0.39) CA1CA2FAAHLMNACYP1A2
SCHEMBL8190241 0.63 CLK4 (0.49) LMNACYP1A2CYP3A4HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020081508-A1 TYK2 INHIBITORS AND USES THEREOF NIMBUS LAKSHMI, INC. (US) 2020-04-23 WO disclosed