SCHEMBL21955474

SCHEMBL21955474

CN(Cc1c(F)ccc(F)c1C=NO)C(C)(C)C

nearest known ligand 0.32

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN8A Q9UQD0 4/20 0.32
SCN1A P35498 3/20 0.32
SCN5A Q14524 3/20 0.32
RIPK1 Q13546 1/20 0.31
HPGD P15428 1/20 0.31
NR1I2 O75469 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
SCN1B Q07699 1/20 0.30
KCNH2 Q12809 1/20 0.30
SCN9A Q15858 1/20 0.30
SCN2A Q99250 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21783392 1.00 SCN8A (0.32) SCN8ASCN1ASCN5ARIPK1HPGD
SCHEMBL22349494 0.84 HPGD (0.33) HPGDCYP3A4
SCHEMBL21783391 0.80 SCN1A (0.33) SCN8ASCN1ASCN5ARIPK1
SCHEMBL22349499 0.74 HPGD (0.41) HPGD
SCHEMBL20238137 0.71 HPGD (0.33) HPGD
SCHEMBL21783477 0.70 SCN1A (0.33) SCN8ASCN1ASCN5ARIPK1
SCHEMBL21783394 0.70 SCN1A (0.35) SCN8ASCN1ASCN5ARIPK1
SCHEMBL22331156 0.70 SCN8A (0.39) SCN8AHPGD
SCHEMBL22096868 0.65 HPGD (0.36) HPGD
SCHEMBL21777310 0.65 ALDH1A1 (0.41) HPGDCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112638879-B Heteroaryl substituted sulfonamide compounds and their use as therapeutic agents 泽农医药公司 2024-06-18 CN disclosed
US-11639351-B2 Heteroaryl-substituted sulfonamide compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC. 2023-05-02 US disclosed
US-11639351-B2 Heteroaryl-substituted sulfonamide compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC. 2023-05-02 US disclosed
US-20220348570-A1 HETEROARYL-SUBSTITUTED SULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2022-11-03 US disclosed
US-10981905-B2 Heteroaryl-substituted sulfonamide compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2021-04-20 US disclosed
CN-112638879-A Heteroaryl substituted sulfonamide compounds and their use as therapeutic agents 泽农医药公司 2021-04-09 CN disclosed
US-20200157089-A1 HETEROARYL-SUBSTITUTED SULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2020-05-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11639351-B2 Heteroaryl-substituted sulfonamide compounds and their use as therapeutic agents SCN1A, SCN2A, SCN2B SCN8A 6/4885SCN1A 1/4885SCN5A 7/4885
US-20200157089-A1 HETEROARYL-SUBSTITUTED SULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS SCN1A, SCN2A, SCN2B SCN8A 6/4885SCN1A 1/4885SCN5A 7/4885
US-10981905-B2 Heteroaryl-substituted sulfonamide compounds and their use as therapeutic agents SCN1A, SCN2A, SCN2B SCN8A 6/4885SCN1A 1/4885SCN5A 7/4885
US-20220348570-A1 HETEROARYL-SUBSTITUTED SULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS SCN1A, SCN2A, SCN2B SCN8A 6/4885SCN1A 1/4885SCN5A 7/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.