SCHEMBL21958702

SCHEMBL21958702

CC1CN(C)CC1Cc1ccccn1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 2/20 0.44
PRKAG1 P54619 2/20 0.44
PRKAA1 Q13131 2/20 0.44
NEK1 Q96PY6 2/20 0.44
PRKAB1 Q9Y478 2/20 0.44
HRH3 Q9Y5N1 3/20 0.43
LMNA P02545 2/20 0.41
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 1/20 0.38
KCNH2 Q12809 1/20 0.38
LTB4R Q15722 1/20 0.37
LTB4R2 Q9NPC1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24780661 0.81 LMNA (0.39) IKBKBPRKAG1PRKAA1NEK1PRKAB1
SCHEMBL8091807 0.80 HRH3 (0.43) HRH3LMNALTB4RLTB4R2
SCHEMBL8094726 0.80 HRH3 (0.43) HRH3LMNALTB4RLTB4R2
SCHEMBL16269835 0.80 HRH3 (0.43) HRH3LMNALTB4RLTB4R2
SCHEMBL25112109 0.75 HRH4 (0.41) IKBKBPRKAG1PRKAA1NEK1PRKAB1
SCHEMBL12090211 0.73 MAP4K4 (0.49) IKBKBPRKAG1PRKAA1NEK1PRKAB1
SCHEMBL9965979 0.73 LMNA (0.48) IKBKBPRKAG1PRKAA1NEK1PRKAB1
SCHEMBL8302404 0.71 KDM4E (0.50) IKBKBPRKAG1PRKAA1NEK1PRKAB1
SCHEMBL12090380 0.71 KCNH2 (0.53) IKBKBPRKAG1PRKAA1NEK1PRKAB1
SCHEMBL25839727 0.71 HRH3 (0.46) IKBKBPRKAG1PRKAA1NEK1PRKAB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020081572-A1 TRANSCRIPTIONAL ENHANCED ASSOCIATE DOMAIN (TEAD) TRANSCRIPTION FACTOR INHIBITORS AND USES THEREOF DANA-FARBER CANCER INSTITUTE, INC. (US) 2020-04-23 WO disclosed