SCHEMBL21962533

SCHEMBL21962533

O=C(c1cccc(C(F)(F)F)c1)c1cnc(N2CC3CC2C3)s1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
MAPT P10636 1/20 0.40
ADORA1 P30542 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CES2 O00748 1/20 0.40
VNN1 O95497 6/20 0.40
CNR2 P34972 2/20 0.39
KCNQ3 O43525 1/20 0.39
KCNQ2 O43526 1/20 0.39
KCNE1 P15382 1/20 0.39
KCNQ1 P51787 1/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21962791 0.93 MEN1 (0.42) SRD5A2MEN1KMT2AALDH1A1CYP1A2
SCHEMBL21962451 0.91 MEN1 (0.41) SRD5A2MEN1KMT2AALDH1A1CYP1A2
SCHEMBL21962579 0.81 SRD5A2 (0.43) SRD5A2MEN1KMT2AALDH1A1CYP1A2
SCHEMBL21962395 0.81 SRD5A2 (0.43) SRD5A2MEN1KMT2AALDH1A1CYP1A2
SCHEMBL22019136 0.81 SRD5A2 (0.43) SRD5A2MEN1KMT2AALDH1A1CYP1A2
SCHEMBL21962600 0.81 HPGD (0.42) SRD5A2MEN1KMT2AALDH1A1CYP1A2
SCHEMBL21962547 0.81 HDAC3 (0.44) SRD5A2MEN1KMT2AALDH1A1CYP1A2
SCHEMBL22020545 0.81 HDAC3 (0.44) SRD5A2MEN1KMT2AALDH1A1CYP1A2
SCHEMBL21962651 0.80 VNN1 (0.43) SRD5A2MEN1KMT2AALDH1A1CYP1A2
SCHEMBL21962779 0.79 MLYCD (0.49) SRD5A2MEN1KMT2AALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102575-A1 HETEROCYCLIC AMINOTHIAZOLES AND USES THEREOF INCEPTION IBD, INC. (US) 2020-05-22 WO claimed
WO-2020102575-A1 HETEROCYCLIC AMINOTHIAZOLES AND USES THEREOF INCEPTION IBD, INC. (US) 2020-05-22 WO disclosed
WO-2020102575-A1 HETEROCYCLIC AMINOTHIAZOLES AND USES THEREOF INCEPTION IBD, INC. (US) 2020-05-22 WO disclosed