Phenyramidol

Phenyramidol

SCHEMBL21963

OC(CNc1ccccn1)c1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 1.00
KDM4E B2RXH2 3/20 0.58
FDPS P14324 1/20 0.55
L3MBTL1 Q9Y468 2/20 0.53
FABP1 P07148 1/20 0.51
FABP6 P51161 1/20 0.51
FAAH O00519 10/20 0.50
AOC3 Q16853 3/20 0.50
CXCR4 P61073 1/20 0.49
HTT P42858 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phenyramidol SCHEMBL13310227 1.00 CYP2D6 (1.00) CYP2D6KDM4EFDPSL3MBTL1FABP1
Phenyramidol SCHEMBL13310219 1.00 CYP2D6 (1.00) CYP2D6KDM4EFDPSL3MBTL1FABP1
Phenyramidol SCHEMBL29500950 1.00 CYP2D6 (1.00) CYP2D6KDM4EFDPSL3MBTL1FABP1
Phenyramidol SCHEMBL20769334 0.98 CYP2D6 (0.97) CYP2D6KDM4EFDPSL3MBTL1FABP1
Phenyramidol SCHEMBL29375712 0.98 CYP2D6 (0.97) CYP2D6KDM4EFDPSL3MBTL1FABP1
Phenyramidol SCHEMBL121004 0.98 CYP2D6 (0.97) CYP2D6KDM4EFDPSL3MBTL1FABP1
Phenyramidol SCHEMBL3446649 0.94 CYP2D6 (0.88) CYP2D6KDM4EFDPSL3MBTL1FABP1
SCHEMBL9566716 0.87 CYP2D6 (0.77) CYP2D6KDM4EFDPSFABP1FABP6
Phenyramidol SCHEMBL22718457 0.84 CYP2D6 (0.71) CYP2D6KDM4EFDPSFAAHAOC3
SCHEMBL4281005 0.84 CYP2D6 (0.72) CYP2D6KDM4EFDPSL3MBTL1FABP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5975 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025062440-A1 TOPICAL NANO-DISPERSION COMPOSITIONS AND THEIR PREPARATION THEREOF PULSE PHARMACEUTICALS PVT. LTD (IN) 2025-03-27 WO claimed
US-20230285282-A1 OCULAR IMPLANT CONTAINING AN ACTIVE INGREDIENT OCULAR THERAPEUTIX INC (US) 2023-09-14 US claimed
EP-4236943-A1 OCULAR IMPLANT CONTAINING AN ACTIVE AGENT Ocular Therapeutix, Inc. (US) 2023-09-06 EP claimed
EP-1931320-B1 MICROPARTICLES WITH MODIFIED RELEASE OF AT LEAST ONE ACTIVE PRINCIPLE AND ORAL DOSAGE FORM COMPRISING THE SAME FLAMEL IRELAND LTD (IE) 2022-06-15 EP claimed
US-20220133616-A1 Compositions, Methods and Uses for Treating Skin Aging EVANS ROBIN JAMES (US) 2022-05-05 US claimed
WO-2022093818-A1 OCULAR IMPLANT CONTAINING AN ACTIVE AGENT OCULAR THERAPEUTIX, INC. (US) 2022-05-05 WO claimed
EP-3797098-A1 SOLID ORAL PHARMACEUTICAL COMPOSITIONS COMPRISING PHENYRAMIDOL OR SALTS THEREOF Santa Farma Ilaç Sanayi A.S. (TR) 2021-03-31 EP claimed
WO-2020101585-A1 SOLID ORAL PHARMACEUTICAL COMPOSITIONS COMPRISING PHENYRAMIDOL OR SALTS THEREOF SANTA FARMA İLAÇ SANAYİ A.Ş. (TR) 2020-05-22 WO claimed
US-20150306063-A1 COMPOSITION AND METHOD FOR VAGINAL THERAPY MCGINNIS DIANE (US) 2015-10-29 US claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
WO-2001012584-A2 PHARMACEUTICAL COMPOUNDS NICOX S.A. (FR) 2001-02-22 WO claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000061541-A2 PHARMACEUTICAL COMPOUNDS NICOX S.A. (FR) 2000-10-19 WO claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
WO-1997020551-A1 PHARMACEUTICAL COMPOSITION COMPRISING A SKELETAL MUSCLE RELAXANT, A NON-STEROIDAL ANTIINFLAMMATORY AGENT AND AN ANALGESIC ADCOCK INGRAM LIMITED (ZA) 1997-06-12 WO claimed
US-4780463-A CONTAINING PROPIONIC ACID COMPOUNDS ANALGESIC ASSOCIATES (US) 1988-10-25 US claimed
US-RE32393-E STABLE, OIL IN WATER EMULSION KABIVITRUM AB (SE) 1987-04-07 US claimed
EP-0205492-A1 ANALGESIC, ANTI-INFLAMMATORY AND SKELETAL MUSCLE RELAXANT COMPOSITIONS SUNSHINE, Abraham (US) 1986-12-30 EP claimed
WO-1986003681-A1 ANALGESIC, ANTI-INFLAMMATORY AND SKELETAL MUSCLE RELAXANT COMPOSITIONS SUNSHINE ABRAHAM 1986-07-03 WO claimed
US-4168308-A Composition for enhancing the administration of pharmacologically active agents APOTEKSVARUCENTRALEN VITRUM AB (SE) 1979-09-18 US claimed