SCHEMBL21968985

SCHEMBL21968985

Cc1cccc(C#Cc2cncc(OCC3CCN3C(=O)OC(C)(C)C)c2)c1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 15/20 0.56
CHRNA4 P43681 8/20 0.56
GRM5 P41594 3/20 0.54
CHRNA3 P32297 7/20 0.49
CHRNB1 P11230 2/20 0.49
CHRNB4 P30926 2/20 0.49
CHRNB3 Q05901 2/20 0.49
CHRNA2 Q15822 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16194566 1.00 CHRNB2 (0.56) CHRNB2CHRNA4GRM5CHRNA3CHRNB1
SCHEMBL21968841 0.91 CHRNB2 (0.65) CHRNB2CHRNA4GRM5CHRNA3CHRNB1
SCHEMBL14941722 0.91 CHRNB2 (0.65) CHRNB2CHRNA4GRM5CHRNA3CHRNB1
SCHEMBL16194984 0.91 CHRNB2 (0.65) CHRNB2CHRNA4GRM5CHRNA3CHRNB1
SCHEMBL21968626 0.90 GRM5 (0.56) CHRNB2CHRNA4GRM5CHRNA3CHRNB1
SCHEMBL21968838 0.90 CHRNB2 (0.55) CHRNB2CHRNA4GRM5CHRNA3CHRNB1
SCHEMBL16194622 0.90 GRM5 (0.56) CHRNB2CHRNA4GRM5CHRNA3CHRNB1
SCHEMBL16194582 0.90 CHRNB2 (0.55) CHRNB2CHRNA4GRM5CHRNA3CHRNB1
SCHEMBL3358853 0.90 CHRNB2 (0.52) CHRNB2CHRNA4GRM5CHRNA3CHRNB1
SCHEMBL14941763 0.89 CHRNB2 (0.58) CHRNB2CHRNA4GRM5CHRNA3CHRNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2776423-B1 PHENYL-SUBSTITUTED NICOTINIC LIGANDS, AND METHODS OF USE THEREOF UNIV GEORGETOWN (US) 2020-05-06 EP disclosed