SCHEMBL21974584

SCHEMBL21974584

C#Cc1cncc(C(CC#N)SC)c1

nearest known ligand 0.32

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.31
CYP2A6 P11509 1/20 0.31
CHRNA1 P02708 3/20 0.31
CHRNB4 P30926 3/20 0.31
CHRNA3 P32297 3/20 0.31
CHRNB2 P17787 2/20 0.31
CHRNA4 P43681 2/20 0.31
CHRNG P07510 1/20 0.31
CHRNB1 P11230 1/20 0.31
CHRND Q07001 1/20 0.31
CHRNA2 Q15822 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19592264 0.88 RAF1 (0.33)
SCHEMBL18600079 0.80 CTSB (0.32)
SCHEMBL171179 0.80 CYP2A6 (0.33) GRM5CYP2A6CHRNA1CHRNB4CHRNA3
SCHEMBL9918235 0.78 GRM5 (0.32) GRM5CYP2A6CHRNA1CHRNB4CHRNA3
SCHEMBL22931080 0.77 CYP2A6 (0.33) GRM5CYP2A6CHRNA1CHRNB4CHRNA3
SCHEMBL19592358 0.77 PBRM1 (0.35) GRM5
SCHEMBL19592420 0.76 CYP19A1 (0.37)
SCHEMBL21975098 0.75 CYP11B1 (0.35)
SCHEMBL13774815 0.74 GRM5 (0.30) GRM5CYP2A6
SCHEMBL12329945 0.74 CTSL (0.32) GRM5CYP2A6CHRNA3CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2343298-B9 Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors INCYTE HOLDINGS CORP (US) 2020-05-06 EP disclosed