SCHEMBL21976306

SCHEMBL21976306

O=C(NO)c1ccc2c(c1)NC(c1ccc(OCCOc3ccccc3)cc1)N2

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 5/20 0.47
PARP10 Q53GL7 1/20 0.47
KDM1A O60341 3/20 0.47
PKM P14618 1/20 0.46
MAPT P10636 1/20 0.45
RAB9A P51151 1/20 0.45
SMPD1 P17405 4/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HDAC8 Q9BY41 1/20 0.42
NPC1 O15118 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21976479 0.91 HDAC6 (0.50) HDAC6PARP10KDM1APKMMAPT
SCHEMBL21976248 0.85 HDAC6 (0.45) HDAC6PARP10KDM1APKMMAPT
SCHEMBL21976492 0.81 SMPD1 (0.53) HDAC6MAPTRAB9ASMPD1MEN1
SCHEMBL21976503 0.74 MEN1 (0.45) HDAC6MAPTMEN1KMT2AHDAC8
SCHEMBL21976308 0.74 HDAC6 (0.51) HDAC6SMPD1MEN1KMT2AHDAC8
SCHEMBL21976251 0.74 HDAC6 (0.52) HDAC6SMPD1HDAC8
SCHEMBL21976229 0.74 GAA (0.46) HDAC6KDM1AMAPTRAB9AMEN1
SCHEMBL21976963 0.72 HDAC6 (0.49) HDAC6SMPD1HDAC8
SCHEMBL21976203 0.72 GAA (0.49) HDAC6MAPTMEN1KMT2AHDAC8
SCHEMBL21976470 0.72 HDAC6 (0.55) HDAC6MEN1KMT2AHDAC8NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3294715-B1 BENZIMIDAZOLE DERIVATES USEFUL AS INHIBITORS OF MAMMALIAN HISTONE DEACETYLASE ACTIVITY KANCERA AB (SE) 2020-05-06 EP disclosed