SCHEMBL21976355

SCHEMBL21976355

CNc1ccc(C(=O)N2CCC(O)(c3cccc(C(F)(F)F)c3)CC2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKLR P30613 2/20 0.61
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
ABCB11 O95342 1/20 0.51
TP53 P04637 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
PKM P14618 1/20 0.51
TSHR P16473 1/20 0.51
MAPK1 P28482 1/20 0.51
THPO P40225 1/20 0.51
MTOR P42345 1/20 0.51
EBP Q15125 1/20 0.51
SIGMAR1 Q99720 1/20 0.51
OPRL1 P41146 7/20 0.50
OPRM1 P35372 6/20 0.50
KDM4E B2RXH2 2/20 0.50
PMP22 Q01453 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
CHRM4 P08173 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14282343 0.85 POLB (0.61) PKLRMEN1KMT2AABCB11TP53
SCHEMBL14282310 0.81 S1PR2 (0.60) PKLRMEN1KMT2AOPRL1OPRM1
SCHEMBL11521599 0.79 PKLR (0.57) PKLRMEN1KMT2AABCB11TP53
SCHEMBL2925749 0.79 OPRM1 (0.63) MEN1KMT2AABCB11TP53CYP3A4
SCHEMBL4186712 0.78 PKLR (0.55) PKLRMEN1KMT2AABCB11TP53
SCHEMBL1760977 0.78 OPRL1 (0.62) MEN1KMT2AABCB11TP53CYP3A4
SCHEMBL21976370 0.77 PKLR (0.71) PKLR
SCHEMBL5912310 0.77 GRIN2B (0.63) OPRL1OPRM1CHRM4LMNA
SCHEMBL28821627 0.77 PKLR (0.49) PKLROPRM1KDM4ERXFP1POLB
SCHEMBL16049680 0.77 PKLR (1.00) PKLR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970189-B1 THERAPEUTIC COMPOUNDS AND COMPOSITIONS AGIOS PHARMACEUTICALS INC (US) 2020-05-06 EP disclosed