SCHEMBL21976964

SCHEMBL21976964

CCCCc1ccc(-c2nc3ccc(C)cc3[nH]2)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MPL P40238 2/20 0.65
HDAC3 O15379 1/20 0.64
HDAC1 Q13547 1/20 0.64
HDAC2 Q92769 1/20 0.64
HDAC8 Q9BY41 1/20 0.64
HDAC6 Q9UBN7 1/20 0.64
NPC1 O15118 2/20 0.59
RAB9A P51151 2/20 0.59
NPBWR1 P48145 2/20 0.56
MMP2 P08253 2/20 0.55
MMP9 P14780 2/20 0.55
MMP8 P22894 2/20 0.55
MMP13 P45452 2/20 0.55
HPSE Q9Y251 1/20 0.54
ACHE P22303 2/20 0.54
ALOX5 P09917 1/20 0.53
EPHX2 P34913 1/20 0.53
PTGDR2 Q9Y5Y4 1/20 0.52
KMT2A Q03164 1/20 0.51
KDM4E B2RXH2 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9295731 0.89 MPL (0.67) MPLHDAC3HDAC1HDAC2HDAC8
SCHEMBL13599850 0.84 NPC1 (0.81) NPC1RAB9ANPBWR1MMP2MMP9
SCHEMBL13183701 0.82 NPC1 (0.78) NPC1RAB9ANPBWR1MMP2MMP9
SCHEMBL9095200 0.82 MPL (0.63) MPLHDAC3HDAC1HDAC2HDAC8
SCHEMBL6544064 0.82 MPL (0.59) MPLHDAC3HDAC1HDAC2HDAC8
SCHEMBL9295738 0.82 MPL (0.48) MPLHDAC3HDAC1HDAC2HDAC8
SCHEMBL9295726 0.80 MPL (0.57) MPLHDAC3HDAC1HDAC2HDAC8
SCHEMBL3546177 0.79 MPL (1.00) MPLHDAC3HDAC1HDAC2HDAC8
SCHEMBL18229675 0.78 HDAC6 (1.00) MPLHDAC3HDAC1HDAC2HDAC8
SCHEMBL6124301 0.78 NPC1 (0.71) NPC1RAB9ANPBWR1MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3294715-B1 BENZIMIDAZOLE DERIVATES USEFUL AS INHIBITORS OF MAMMALIAN HISTONE DEACETYLASE ACTIVITY KANCERA AB (SE) 2020-05-06 EP disclosed