SCHEMBL21979523

SCHEMBL21979523

CN[C@H](C(=O)Nc1ccc(-c2cn[nH]c2)cc1)c1ccc(Cl)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 20/20 1.00
ROCK1 Q13464 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20661019 1.00 ROCK2 (1.00) ROCK2ROCK1
SCHEMBL20661144 1.00 ROCK2 (1.00) ROCK2ROCK1
SCHEMBL20661152 0.89 ROCK2 (1.00) ROCK2ROCK1
SCHEMBL20661129 0.88 ROCK2 (1.00) ROCK2ROCK1
SCHEMBL20661120 0.88 ROCK2 (1.00) ROCK2ROCK1
SCHEMBL20661139 0.87 ROCK2 (1.00) ROCK2ROCK1
SCHEMBL20661093 0.87 ROCK2 (1.00) ROCK2ROCK1
SCHEMBL20661091 0.86 ROCK2 (1.00) ROCK2ROCK1
SCHEMBL20661029 0.86 ROCK2 (1.00) ROCK2ROCK1
SCHEMBL20661173 0.86 ROCK2 (1.00) ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11479533-B2 Inhibitors of Rho associated coiled-coil containing protein kinase KADMON CORPORATION, LLC (US) 2022-10-25 US disclosed
US-20200165206-A1 INHIBITORS OF RHO ASSOCIATED COILED-COIL CONTAINING PROTEIN KINASE KADMON CORPORATION, LLC 2020-05-28 US disclosed
US-20200165206-A1 INHIBITORS OF RHO ASSOCIATED COILED-COIL CONTAINING PROTEIN KINASE KADMON CORPORATION, LLC 2020-05-28 US disclosed
CN-111050766-A RHO-related inhibitors of coiled-coil protein kinase 卡德门企业有限公司 2020-04-21 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11479533-B2 Inhibitors of Rho associated coiled-coil containing protein kinase ROCK1, ROCK2, RHOT2 ROCK2 2/4885ROCK1 1/4885
US-20200165206-A1 INHIBITORS OF RHO ASSOCIATED COILED-COIL CONTAINING PROTEIN KINASE ROCK1, ROCK2, RHOT2 ROCK2 2/4885ROCK1 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.