SCHEMBL21985657

SCHEMBL21985657

C=C(C)C1=CC=C(C(=O)O)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.43
LMNA P02545 2/20 0.43
CES2 O00748 3/20 0.36
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB1 P18505 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRR1 P24046 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA5 P31644 1/20 0.33
GABRA3 P34903 1/20 0.33
GABRA2 P47869 1/20 0.33
GABRB2 P47870 1/20 0.33
GABRA4 P48169 1/20 0.33
GABRE P78334 1/20 0.33
GABRA6 Q16445 1/20 0.33
GABRG1 Q8N1C3 1/20 0.33
GABRG3 Q99928 1/20 0.33
GABRQ Q9UN88 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1355407 0.83 TSHR (0.42) TSHRLMNACES2GABRPGABRD
Benzene SCHEMBL11562666 0.76 LMNA (0.31) LMNA
SCHEMBL17993483 0.74 TSHR (0.34) TSHRLMNACES2GABRPGABRD
SCHEMBL23067733 0.74 LMNA (0.32) LMNA
SCHEMBL14010784 0.71 FFAR1 (0.33) TSHRLMNACES2GABRPGABRD
SCHEMBL21291247 0.71 LMNA (0.32) TSHRLMNA
SCHEMBL23864852 0.71 KDM4E (0.38) TSHRLMNABLMMAPK1HSD17B10
SCHEMBL24755662 0.70 TSHR (0.34) TSHRLMNAGABRPGABRDGABRA1
SCHEMBL21264412 0.70 TSHR (0.34) TSHRLMNAGABRPGABRDGABRA1
SCHEMBL23300034 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3087060-B1 PYRIMIDONE CARBOXAMIDE COMPOUNDS AS PDE2 INHIBITORS MERCK SHARP & DOHME (US) 2020-05-13 EP disclosed