SCHEMBL21986319

SCHEMBL21986319

Cc1ncc(I)c2nccn12

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2E1 P05181 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2A6 P11509 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.33
LMNA P02545 1/20 0.33
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
KMT2A Q03164 1/20 0.32
FLT1 P17948 1/20 0.31
CDK8 P49336 1/20 0.31
CDK9 P50750 1/20 0.31
LIMK1 P53667 1/20 0.31
ROCK1 Q13464 1/20 0.31
CLK4 Q9HAZ1 1/20 0.31
IKBKB O14920 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14793698 0.79 L3MBTL1 (0.36) CYP2E1CYP3A4CYP2A6L3MBTL1LMNA
SCHEMBL21287497 0.76 AXL (0.32) L3MBTL1
SCHEMBL1685158 0.76 CCNE1 (0.33)
SCHEMBL22521326 0.76 ADORA2A (0.39)
SCHEMBL21287178 0.76 CCNE1 (0.34)
SCHEMBL23709296 0.72 EED (0.40)
SCHEMBL10831370 0.72 KDM4E (0.37) L3MBTL1LMNAALDH1A1KMT2A
SCHEMBL21287821 0.71 HRH4 (0.33) LMNAPOLB
Bromide SCHEMBL10831260 0.71 TLR7 (0.32) L3MBTL1LMNA
SCHEMBL22447092 0.70 EED (0.38) ALDH1A1LIMK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3172214-B1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE DERIVATIVES AS CDK INHIBITORS AND USES THEREOF SUNSHINE LAKE PHARMA CO LTD (CN) 2020-05-13 EP disclosed