SCHEMBL21993350

SCHEMBL21993350

CN(C(=O)C(Cc1cc(F)cc(F)c1)N(C)C(=O)OC(C)(C)C)c1ccc(C2CC2)cc1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
STAT3 P40763 3/20 0.35
POLQ O75417 1/20 0.34
AAK1 Q2M2I8 2/20 0.34
ADORA1 P30542 1/20 0.33
STAT5B P51692 1/20 0.32
USP30 Q70CQ3 2/20 0.32
PER2 O15055 1/20 0.32
CRY1 Q16526 1/20 0.32
CRY2 Q49AN0 1/20 0.32
BACE1 P56817 4/20 0.31
CTSD P07339 3/20 0.31
KDM1A O60341 3/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
PAX8 Q06710 1/20 0.31
IDH1 O75874 1/20 0.31
MAOA P21397 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18180346 0.86 USP30 (0.33) AAK1ADORA1USP30BACE1PAX8
SCHEMBL18180211 0.82 KDM1A (0.45) KDM1AMAOA
SCHEMBL18180190 0.80 AAK1 (0.34) AAK1ADORA1USP30BACE1CTSD
SCHEMBL21993352 0.80 AAK1 (0.34) AAK1ADORA1USP30BACE1CTSD
SCHEMBL21992548 0.79 HDAC1 (0.35) AAK1ADORA1HDAC8HDAC6PAX8
SCHEMBL21992122 0.78 POLQ (0.38) POLQAAK1ADORA1BACE1CTSD
SCHEMBL18180021 0.78 DPP4 (0.38) STAT3POLQPER2CRY1CRY2
SCHEMBL21993354 0.77 AAK1 (0.32) AAK1ADORA1
SCHEMBL21992663 0.76 ADORA1 (0.33) AAK1ADORA1PAX8
SCHEMBL21992323 0.76 AAK1 (0.36) AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3286166-B1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV HEALTHCARE UK NO 5 LTD (GB) 2020-05-13 EP disclosed