SCHEMBL21993352

SCHEMBL21993352

Cc1ccc(N(C)C(=O)C(Cc2cc(F)cc(F)c2)N(C)C(=O)OC(C)(C)C)cn1

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 4/20 0.34
P2RX3 P56373 1/20 0.33
ADORA1 P30542 1/20 0.33
OXTR P30559 2/20 0.32
AVPR1A P37288 1/20 0.32
BACE1 P56817 2/20 0.32
HDAC1 Q13547 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
PAX8 Q06710 1/20 0.31
MAOB P27338 1/20 0.31
REN P00797 1/20 0.31
CTSS P25774 1/20 0.31
CTSK P43235 1/20 0.31
USP30 Q70CQ3 1/20 0.30
MMP13 P45452 1/20 0.30
KCNQ4 P56696 1/20 0.30
KCNQ5 Q9NR82 1/20 0.30
CTSD P07339 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18180190 1.00 AAK1 (0.34) AAK1P2RX3ADORA1OXTRAVPR1A
SCHEMBL21992548 0.89 HDAC1 (0.35) AAK1P2RX3ADORA1HDAC1HDAC8
SCHEMBL21992122 0.86 POLQ (0.38) AAK1ADORA1BACE1RENMMP13
SCHEMBL21993354 0.86 AAK1 (0.32) AAK1P2RX3ADORA1
SCHEMBL18180346 0.86 USP30 (0.33) AAK1ADORA1BACE1PAX8USP30
SCHEMBL18181342 0.82 CTSS (0.46) CTSSCTSK
SCHEMBL21993350 0.80 STAT3 (0.35) AAK1ADORA1BACE1HDAC8HDAC6
SCHEMBL21992592 0.80 KMT2A (0.35) AAK1ADORA1HDAC1HDAC8PAX8
SCHEMBL21993353 0.78 ADORA1 (0.30) AAK1ADORA1BACE1
SCHEMBL21993358 0.78 PAX8 (0.39) AAK1ADORA1PAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3286166-B1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV HEALTHCARE UK NO 5 LTD (GB) 2020-05-13 EP disclosed