SCHEMBL21992663

SCHEMBL21992663

CN(C(=O)C(Cc1cc(F)cc(F)c1)N(C)C(=O)OC(C)(C)C)c1ccc2sc(=O)[nH]c2c1

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.33
PAX8 Q06710 1/20 0.32
AAK1 Q2M2I8 2/20 0.31
CMA1 P23946 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18180242 0.84 CTSS (0.41)
SCHEMBL21993358 0.81 PAX8 (0.39) ADORA1PAX8AAK1
SCHEMBL18180050 0.80 CMA1 (0.35) CMA1
SCHEMBL18180190 0.76 AAK1 (0.34) ADORA1PAX8AAK1
SCHEMBL21993350 0.76 STAT3 (0.35) ADORA1PAX8AAK1
SCHEMBL21993352 0.76 AAK1 (0.34) ADORA1PAX8AAK1
SCHEMBL21992548 0.75 HDAC1 (0.35) ADORA1PAX8AAK1
SCHEMBL21992122 0.74 POLQ (0.38) ADORA1AAK1
SCHEMBL21992592 0.74 KMT2A (0.35) ADORA1PAX8AAK1
SCHEMBL21992323 0.74 AAK1 (0.36) AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3286166-B1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV HEALTHCARE UK NO 5 LTD (GB) 2020-05-13 EP disclosed