SCHEMBL21994256

SCHEMBL21994256

COc1ccc(CC(=O)NC2CNCC2c2ccc(C(F)(F)F)cc2)cn1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.65
CYP3A4 P08684 3/20 0.65
CYP2D6 P10635 3/20 0.65
CYP2C19 P33261 3/20 0.65
CYP2C9 P11712 2/20 0.65
AKT1 P31749 3/20 0.46
MAPK1 P28482 1/20 0.44
PRKAA2 P54646 5/20 0.41
PIK3CA P42336 4/20 0.41
PRKAB2 O43741 2/20 0.41
PRKAG1 P54619 2/20 0.41
PRKAA1 Q13131 2/20 0.41
PRKAG3 Q9UGI9 2/20 0.41
PRKAG2 Q9UGJ0 2/20 0.41
PRKAB1 Q9Y478 2/20 0.41
KDM1A O60341 1/20 0.40
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
CCNE1 P24864 2/20 0.40
CDK2 P24941 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21994286 0.87 KCNH2 (0.68) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994254 0.85 KCNH2 (0.74) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994284 0.81 KCNH2 (0.78) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994263 0.81 KCNH2 (0.57) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994259 0.80 KCNH2 (0.63) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994288 0.79 KCNH2 (0.75) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994243 0.79 KCNH2 (0.74) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994246 0.79 KCNH2 (0.74) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994239 0.79 KCNH2 (1.00) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994242 0.76 KCNH2 (0.67) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020107189-A1 PYRROLIDINE COMPOUNDS FOR THE TREATMENT OF MALARIA LEGION PHARMA CO. LTD (CN) 2020-06-04 WO claimed