SCHEMBL21994263

SCHEMBL21994263

COc1ccc(CC(=O)NC2CNCC2c2ccc(C(F)(F)F)cc2)nc1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.57
CYP3A4 P08684 3/20 0.57
CYP2D6 P10635 3/20 0.57
CYP2C19 P33261 3/20 0.57
CYP2C9 P11712 2/20 0.57
AKT1 P31749 3/20 0.44
MAPK1 P28482 1/20 0.44
RPS6KB1 P23443 1/20 0.39
TP53 P04637 1/20 0.39
CCNE1 P24864 2/20 0.39
CDK2 P24941 2/20 0.39
GSK3B P49841 2/20 0.39
DGAT2 Q96PD7 1/20 0.38
FPR1 P21462 2/20 0.38
MAPT P10636 1/20 0.38
ROCK2 O75116 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21994254 0.85 KCNH2 (0.74) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994256 0.81 KCNH2 (0.65) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994259 0.80 KCNH2 (0.63) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994286 0.77 KCNH2 (0.68) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994284 0.75 KCNH2 (0.78) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994243 0.75 KCNH2 (0.74) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994288 0.73 KCNH2 (0.75) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994239 0.73 KCNH2 (1.00) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994246 0.73 KCNH2 (0.74) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994242 0.72 KCNH2 (0.67) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020107189-A1 PYRROLIDINE COMPOUNDS FOR THE TREATMENT OF MALARIA LEGION PHARMA CO. LTD (CN) 2020-06-04 WO claimed