SCHEMBL21996281

SCHEMBL21996281

[CH2]c1ccc(CNC(=O)OC(C)(C)C)c(F)c1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 3/20 0.43
NR1H4 Q96RI1 2/20 0.43
KDM4A O75164 1/20 0.43
KCNA5 P22460 1/20 0.40
BDKRB1 P46663 4/20 0.39
RIPK1 Q13546 1/20 0.39
IDO1 P14902 2/20 0.38
NQO2 P16083 1/20 0.38
GRM2 Q14416 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
RPS6KA1 Q15418 1/20 0.37
CACNA1H O95180 1/20 0.37
CACNA1B Q00975 1/20 0.37
CACNA1C Q13936 1/20 0.37
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12791296 0.86 P2RX7 (0.46) EPHX2NR1H4KDM4AKCNA5BDKRB1
SCHEMBL4894133 0.84 NQO2 (0.49) EPHX2NR1H4KDM4AKCNA5BDKRB1
SCHEMBL506329 0.83 AAK1 (0.50) EPHX2NR1H4KDM4ABDKRB1
SCHEMBL4597727 0.83 AKR1B1 (0.46) EPHX2NR1H4KDM4AKCNA5BDKRB1
SCHEMBL24791641 0.83 EPHX2 (0.43) EPHX2NR1H4KDM4AKCNA5BDKRB1
SCHEMBL30193009 0.83 EPHX2 (0.49) EPHX2NR1H4KDM4AKCNA5BDKRB1
SCHEMBL23832914 0.83 EPHX2 (0.49) EPHX2NR1H4KDM4AKCNA5BDKRB1
SCHEMBL26828546 0.82 EPHX2 (0.42) EPHX2NR1H4KDM4AKCNA5BDKRB1
SCHEMBL12231326 0.82 GRM2 (0.43) EPHX2NR1H4KDM4AKCNA5BDKRB1
SCHEMBL1495902 0.82 EPHX2 (0.64) EPHX2NR1H4KDM4AKCNA5BDKRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3886854-A1 PYRROLE AND PYRAZOLE COMPOUNDS AND METHODS OF USE THEREOF Nuvation Bio Inc. (US) 2021-10-06 EP disclosed
WO-2020113094-A1 PYRROLE AND PYRAZOLE COMPOUNDS AND METHODS OF USE THEREOF NUVATION BIO INC. (US) 2020-06-04 WO disclosed