SCHEMBL21996596

SCHEMBL21996596

COC(=O)C1CC(OCc2cc(F)c(F)c(F)c2)CN1C(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 2/20 0.42
PTPN1 P18031 1/20 0.40
ABCB1 P08183 1/20 0.39
NR1H2 P55055 1/20 0.38
NR1H3 Q13133 1/20 0.38
CYP1A2 P05177 1/20 0.36
POLB P06746 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
BACE1 P56817 2/20 0.36
BACE2 Q9Y5Z0 1/20 0.36
UCHL1 P09936 1/20 0.35
CCNT1 O60563 1/20 0.35
CDK9 P50750 1/20 0.35
MCL1 Q07820 2/20 0.34
DRD4 P21917 1/20 0.34
TMEM97 Q5BJF2 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
CETP P11597 1/20 0.34
KLK7 P49862 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21996539 0.86 P2RX3 (0.44) P2RX3PTPN1ABCB1NR1H2NR1H3
SCHEMBL15499687 0.85 ABCB1 (0.42) P2RX3ABCB1NR1H2NR1H3BACE1
SCHEMBL475486 0.84 ABCB1 (0.52) P2RX3ABCB1NR1H2NR1H3UCHL1
SCHEMBL3854950 0.84 ABCB1 (0.52) P2RX3ABCB1NR1H2NR1H3UCHL1
SCHEMBL3191348 0.84 ABCB1 (0.52) P2RX3ABCB1NR1H2NR1H3UCHL1
SCHEMBL18093988 0.84 ABCB1 (0.52) P2RX3ABCB1NR1H2NR1H3UCHL1
SCHEMBL475487 0.84 ABCB1 (0.52) P2RX3ABCB1NR1H2NR1H3UCHL1
SCHEMBL21996445 0.83 ABCB1 (0.43) ABCB1NR1H2BACE1BACE2GPR119
SCHEMBL3857592 0.82 P2RX3 (0.48) P2RX3ABCB1CYP3A4MCL1GPR119
SCHEMBL3190398 0.82 P2RX3 (0.54) P2RX3ABCB1NR1H2NR1H3CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020113077-A9 COMPOSITIONS AND METHODS FOR MODULAR CONTROL OF BIOORTHOGONAL LIGATION THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2020-08-13 WO disclosed
WO-2020113077-A1 COMPOSITIONS AND METHODS FOR MODULAR CONTROL OF BIOORTHOGONAL LIGATION THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2020-06-04 WO disclosed
WO-2020113077-A1 COMPOSITIONS AND METHODS FOR MODULAR CONTROL OF BIOORTHOGONAL LIGATION THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2020-06-04 WO disclosed