SCHEMBL22005771

SCHEMBL22005771

CN1C(=O)NCOCC(N2C(=O)c3ccccc3C2=O)C1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 7/20 0.41
CRBN Q96SW2 7/20 0.41
CYP1A2 P05177 2/20 0.41
IKZF3 Q9UKT9 2/20 0.41
ALDH1A1 P00352 1/20 0.41
CHRM2 P08172 1/20 0.41
OPRM1 P35372 1/20 0.41
TSHR P16473 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CASP3 P42574 1/20 0.39
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.33
NR1H3 Q13133 4/20 0.33
NR1H2 P55055 2/20 0.33
TNF P01375 1/20 0.33
IL1B P01584 1/20 0.33
TBXA2R P21731 1/20 0.33
IKZF1 Q13422 1/20 0.33
TTR P02766 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20046006 0.81 CRBN (0.46) DDB1CRBNCYP1A2IKZF3ALDH1A1
SCHEMBL30250317 0.72 RIPK1 (0.49)
SCHEMBL845548 0.69 CRBN (0.54) DDB1CRBNCYP1A2IKZF3ALDH1A1
SCHEMBL2188355 0.67 CRBN (0.47) DDB1CRBNCYP1A2IKZF3ALDH1A1
SCHEMBL30250477 0.67 RIPK1 (0.41) DDB1CRBN
SCHEMBL12809078 0.67 CRBN (0.51) DDB1CRBNCYP1A2IKZF3ALDH1A1
SCHEMBL7346208 0.65 CRBN (0.57) DDB1CRBNCYP1A2IKZF3ALDH1A1
SCHEMBL22502405 0.65 CRBN (0.57) DDB1CRBNCYP1A2IKZF3ALDH1A1
SCHEMBL22151223 0.65 CRBN (0.46) CRBNALDH1A1TSHRTDP1L3MBTL1
SCHEMBL31013861 0.65 CRBN (0.49) DDB1CRBNCYP1A2IKZF3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200155690-A1 CEREBLON LIGANDS AND BIFUNCTIONAL COMPOUNDS COMPRISING THE SAME ARVINAS OPERATIONS, INC. 2020-05-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200155690-A1 CEREBLON LIGANDS AND BIFUNCTIONAL COMPOUNDS COMPRISING THE SAME CRBN, CBL, MDM2 DDB1 399/4885CRBN 1/4885CYP1A2 4681/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.