SCHEMBL220090

SCHEMBL220090

c1cc2ncncc2nn1

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.40
RPS6KA5 O75582 1/20 0.30
RPS6KA4 O75676 1/20 0.30
HSP90AA1 P07900 1/20 0.30
PIK3CD O00329 1/20 0.30
PIK3CA P42336 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyrrole SCHEMBL82930 0.87 EGFR (0.36) EGFR
SCHEMBL16878146 0.82 EGFR (0.33) EGFRHSP90AA1
SCHEMBL1263213 0.73 EGFR (0.33) EGFRHSP90AA1
Quinoxaline SCHEMBL23530618 0.72 EGFR (0.62) EGFRPIK3CDPIK3CA
Quinazoline SCHEMBL2726373 0.71 EGFR (0.69) EGFRPIK3CDPIK3CA
SCHEMBL219949 0.71 PKM (0.33)
SCHEMBL127479 0.71 EGFR (0.50) EGFRRPS6KA5RPS6KA4HSP90AA1PIK3CD
SCHEMBL374489 0.70 EGFR (0.37) EGFR
SCHEMBL51486 0.70 EGFR (0.52) EGFRRPS6KA5PIK3CDPIK3CA
SCHEMBL30148832 0.70 EGFR (0.37) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 241 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240246959-A1 BENZIMIDAZOLE DERIVATIVE AND PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF SHENZHEN SALUBRIS PHARMACEUTICALS CO., LTD. (CN) 2024-07-25 US claimed
EP-4242202-A1 BENZIMIDAZOLE DERIVATIVE AND PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF Shenzhen Salubris Pharmaceuticals Co., Ltd. (CN) 2023-09-13 EP claimed
CN-115515956-A Benzimidazole derivative and preparation method and medical application thereof 深圳信立泰药业股份有限公司 2022-12-23 CN claimed
CN-114763352-A GLP-1 receptor agonist and application thereof in medicine 海思科医药集团股份有限公司 2022-07-19 CN claimed
WO-2022111624-A1 BENZIMIDAZOLE DERIVATIVE AND PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 深圳信立泰药业股份有限公司 2022-06-02 WO claimed
WO-2022068772-A1 BENZIMIDAZOLE DERIVATIVE, AND PREPARATION METHOD THEREFOR, AND MEDICAL USE THEREOF 深圳信立泰药业股份有限公司 2022-04-07 WO claimed
EP-2336315-B1 Enzymatic encoding methods for efficient synthesis of large libraries NUEVOLUTION AS (DK) 2017-07-19 EP claimed
EP-2336315-A2 Enzymatic encoding methods for efficient synthesis of large libraries Nuevolution A/S (DK) 2011-06-22 EP claimed
CN-1812792-A Use of dipyridamole or mopidamole for the treatment and prevention of thromboembolic diseases and disorders due to overproduction of thrombin and/or increased thrombin receptor expression BOEHRINGER INGELHEIM INT (DE) 2006-08-02 CN claimed
US-4226863-A BACTERICIDES, ANTIBIOTICS SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1980-10-07 US claimed
US-4125611-A MICROBIOCIDES SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1978-11-14 US claimed
JP-52027794-A None JP disclosed
WO-2025050846-A1 COMPOUND, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND USE THEREOF 中山优理生物医药有限公司 2025-03-13 WO disclosed
EP-4219463-B1 TERPYRIDINE DIKETONE COMPOUND OR SALT THEREOF, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF SHENZHEN SALUBRIS PHARM CO LTD (CN) 2025-01-15 EP disclosed
CN-115594669-B Parallel ring derivative and preparation method and medical application thereof 深圳信立泰药业股份有限公司 2024-11-05 CN disclosed
EP-0414386-A1 Condensed pyrimidine derivates DowElanco (US) 1991-02-27 EP disclosed
EP-0000382-B1 PYRIMIDO (4,5-C)PYRIDAZINES, COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION THE WELLCOME FOUNDATION LIMITED (GB) 1982-10-06 EP disclosed
US-4226863-A BACTERICIDES, ANTIBIOTICS SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1980-10-07 US disclosed
US-4125611-A MICROBIOCIDES SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1978-11-14 US disclosed
JP-S5227794-A PREPARATION OF SYNTHESIS OF NNACYLAMINOO ARYLACETAMIDO CEPHALOSPORIN S SUMITOMO CHEM CO LTD 1977-03-02 JP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240246959-A1 BENZIMIDAZOLE DERIVATIVE AND PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF GLP1R, GIPR, GCGR EGFR 1993/4885RPS6KA5 3345/4885RPS6KA4 3117/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.