SCHEMBL2200934

SCHEMBL2200934

Cc1cc(-n2cnc3cccnc32)ccc1CC(=O)Nc1ccc(OC2CCN(C)CC2)c(C(F)(F)F)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 3/20 0.45
KDR P35968 2/20 0.45
ABL1 P00519 7/20 0.44
RAF1 P04049 2/20 0.44
ARAF P10398 2/20 0.44
KIT P10721 4/20 0.43
MAPK14 Q16539 1/20 0.42
RORC P51449 1/20 0.42
ROCK2 O75116 1/20 0.41
LCK P06239 1/20 0.41
CSF1R P07333 1/20 0.41
PDGFRB P09619 1/20 0.41
BLK P51451 1/20 0.41
DDR1 Q08345 1/20 0.41
DDR2 Q16832 1/20 0.41
FGFR1 P11362 1/20 0.41
NEK2 P51955 4/20 0.39
PLK1 P53350 3/20 0.39
SCD O00767 2/20 0.39
SRC P12931 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2204009 0.92 ROCK2 (0.45) BRAFKDRABL1RAF1ARAF
SCHEMBL2203641 0.90 RORC (0.51) BRAFKDRABL1RAF1ARAF
SCHEMBL2201474 0.88 ABL1 (0.41) BRAFKDRABL1KITDDR1
SCHEMBL2202608 0.86 CSF1R (0.45) BRAFKDRROCK2LCKCSF1R
SCHEMBL1408637 0.85 ABL1 (0.54) BRAFABL1KITCSF1RSRC
SCHEMBL2493761 0.82 ABL1 (0.46) BRAFABL1KITSRC
SCHEMBL1408446 0.81 RET (0.48) KDR
SCHEMBL1414442 0.81 MKNK2 (0.53) KDRABL1SRC
SCHEMBL2204785 0.81 MAPT (0.38)
SCHEMBL2202471 0.80 KDR (0.44) BRAFKDRABL1RORCDDR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7977338-B2 Phenylacetamides being FLT3 inhibitors NOVARTIS AG (CH) 2011-07-12 US claimed
US-20100075980-A1 Phenylacetamides being FLT3 Inhibitors NOVARTIS AG (CH) 2010-03-25 US claimed
US-7977338-B2 Phenylacetamides being FLT3 inhibitors NOVARTIS AG (CH) 2011-07-12 US disclosed
US-20100075980-A1 Phenylacetamides being FLT3 Inhibitors NOVARTIS AG (CH) 2010-03-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100075980-A1 Phenylacetamides being FLT3 Inhibitors FLT3, JAK2, ABL1 BRAF 4/4885KDR 110/4885ABL1 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.