SCHEMBL22012206

SCHEMBL22012206

CC(=O)Nc1c(C(C)C)cc(C#N)cc1C(C)C

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.46
GPR35 Q9HC97 5/20 0.39
DYRK1A Q13627 1/20 0.38
KDM1A O60341 1/20 0.37
MAPK8 P45983 2/20 0.37
MAPK9 P45984 2/20 0.37
IDO1 P14902 1/20 0.36
KMT2A Q03164 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
LMNA P02545 1/20 0.36
ALDH1A1 P00352 2/20 0.36
LRRK2 Q5S007 1/20 0.36
EGFR P00533 1/20 0.35
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
HPGD P15428 1/20 0.34
CYP2C19 P33261 1/20 0.34
RAB9A P51151 1/20 0.34
NLRP3 Q96P20 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22002744 0.85 GPR35 (0.38) GAAGPR35KMT2ASMN1; SMN2LMNA
SCHEMBL22002790 0.81 GPR35 (0.36) GAAGPR35KMT2ASMN1; SMN2LMNA
SCHEMBL22002677 0.81 GPR35 (0.36) GAAGPR35KMT2ASMN1; SMN2LMNA
SCHEMBL22002746 0.80 ABL1 (0.40) GPR35MAPK8MAPK9ALDH1A1NLRP3
SCHEMBL7403709 0.79 DYRK1A (0.45) GAADYRK1AKDM1AIDO1KMT2A
SCHEMBL27419002 0.78 FABP3 (0.52) GAAKMT2ASMN1; SMN2LMNAALDH1A1
SCHEMBL13592557 0.78 GAA (0.52) GAAKMT2ASMN1; SMN2LMNAALDH1A1
SCHEMBL22430585 0.77 HPGD (0.47) GPR35DYRK1AKDM1AIDO1SMN1; SMN2
SCHEMBL20915178 0.77 GAA (0.50) GAAKMT2ASMN1; SMN2LMNAALDH1A1
SCHEMBL22868230 0.76 TTR (0.31) GPR35

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102576-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS INFLAMMASOME RESEARCH, INC. (US) 2020-05-22 WO disclosed