SCHEMBL22012518

SCHEMBL22012518

Cc1ccc(CN(C)C2CCC2)cc1F

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.54
HRH4 Q9H3N8 1/20 0.54
PARP1 P09874 2/20 0.41
SLC6A2 P23975 4/20 0.40
SLC6A4 P31645 4/20 0.40
SLC6A3 Q01959 4/20 0.40
LTA4H P09960 1/20 0.39
ALDH1A1 P00352 2/20 0.38
GRIN2B Q13224 1/20 0.38
DPP4 P27487 2/20 0.37
DPP9 Q86TI2 2/20 0.37
DPP7 Q9UHL4 2/20 0.37
TP53 P04637 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ABCB11 O95342 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
AR P10275 1/20 0.35
CYP2D6 P10635 1/20 0.35
PDE4A P27815 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21962214 0.78 HRH3 (0.48) HRH3HRH4PARP1SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL11688138 0.77 HRH3 (0.58) HRH3HRH4PARP1SLC6A2SLC6A4
SCHEMBL8251603 0.77 HRH3 (0.46) HRH3PARP1SLC6A2SLC6A4ALDH1A1
SCHEMBL22013710 0.76 HRH3 (0.46) HRH3HRH4PARP1SLC6A2SLC6A4
SCHEMBL4517897 0.75 HRH3 (0.47) HRH3HRH4PARP1SLC6A2SLC6A4
SCHEMBL29957867 0.75 HRH3 (0.55) HRH3HRH4PARP1SLC6A2SLC6A4
SCHEMBL12084399 0.74 HRH3 (0.73) HRH3HRH4PARP1SLC6A2SLC6A4
SCHEMBL12082363 0.73 HRH3 (0.77) HRH3HRH4PARP1SLC6A2SLC6A4
SCHEMBL4509098 0.72 HRH3 (0.44) HRH3HRH4PARP1SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL11684009 0.72 ALDH1A1 (0.59) HRH3HRH4PARP1ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102576-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS INFLAMMASOME RESEARCH, INC. (US) 2020-05-22 WO disclosed