SCHEMBL2201273

SCHEMBL2201273

Cc1nnc(N2CCCC(NC(=O)O)C2)n(Cc2cc(F)ccc2C#N)c1=O

nearest known ligand 0.76

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 20/20 0.76
CYP3A4 P08684 1/20 0.51
KCNH2 Q12809 1/20 0.49
FAP Q12884 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2022446 0.90 DPP4 (0.69) DPP4FAP
SCHEMBL2022448 0.90 DPP4 (0.69) DPP4FAP
SCHEMBL2181463 0.89 DPP4 (0.61) DPP4CYP3A4
SCHEMBL2201252 0.87 DPP4 (0.57) DPP4CYP3A4FAP
SCHEMBL2200504 0.87 DPP4 (0.57) DPP4CYP3A4FAP
SCHEMBL2020372 0.86 DPP4 (1.00) DPP4KCNH2FAP
SCHEMBL2020371 0.86 DPP4 (1.00) DPP4KCNH2FAP
Benzoic Acid SCHEMBL28645610 0.84 DPP4 (1.00) DPP4CYP3A4KCNH2FAP
SCHEMBL28636345 0.84 DPP4 (0.76) DPP4KCNH2FAP
SCHEMBL28461817 0.81 DPP4 (0.60) DPP4CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2521721-A1 3-(3-AMINOPIPERIDIN-1-YL)-5-OXO-1,2,4-TRIAZINE DERIVATES AS DIPEPTIDYL PEPTIDASE IV(DPP-IV) INHIBITORS Shanghai Fochon Pharmaceutical Co. Ltd (CN) 2012-11-14 EP disclosed
WO-2011079778-A1 3-(3-AMINOPIPERIDIN-1-YL)-5-OXO-1,2,4-TRIAZINE DERIVATES AS DIPEPTIDYL PEPTIDASE IV(DPP-IV) INHIBITORS CHINA SHANGHAI FOCHON PHARMACEUTICAL CO LTD (CN) 2011-07-07 WO disclosed