SCHEMBL22013198

SCHEMBL22013198

CC(=O)NC(=O)c1sc(-c2ccccc2)cc1C=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.51
MAPT P10636 4/20 0.51
ALDH1A1 P00352 3/20 0.51
LMNA P02545 2/20 0.51
PKM P14618 1/20 0.48
RXFP1 Q9HBX9 1/20 0.48
HPGD P15428 2/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
IKBKB O14920 4/20 0.45
NPSR1 Q6W5P4 1/20 0.43
NQO2 P16083 1/20 0.43
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
BTK Q06187 1/20 0.42
MAPK1 P28482 1/20 0.42
APOBEC3A P31941 1/20 0.42
APOBEC3G Q9HC16 1/20 0.42
PTPRF P10586 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12409619 0.81 PTPRF (0.53) KDM4EMAPTALDH1A1LMNAPKM
SCHEMBL2157737 0.74 MAPT (0.44) KDM4EMAPTALDH1A1LMNAPKM
SCHEMBL3102075 0.71 RAB9A (0.46) KDM4EMAPTALDH1A1LMNAPKM
SCHEMBL12987243 0.71 MAPT (0.42) KDM4EMAPTALDH1A1LMNAPKM
SCHEMBL15573218 0.69 RAB9A (0.44) KDM4EMAPTALDH1A1LMNAPKM
SCHEMBL6348871 0.68 PTPN1 (0.56) KDM4EMAPTMEN1KMT2AIKBKB
SCHEMBL3600422 0.68 PTPN1 (0.56) KDM4EMAPTALDH1A1MEN1KMT2A
SCHEMBL5368759 0.68 MAPT (1.00) KDM4EMAPTALDH1A1LMNAHPGD
SCHEMBL16750169 0.67 GAA (0.54) KDM4EMAPTALDH1A1LMNAPKM
SCHEMBL17226314 0.67 PTPN1 (0.68) KDM4EMAPTALDH1A1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102243-A2 IN-FLOW PHOTOOXYGENATION OF AMINOTHIENOPYRIDINONES GENERATES NOVEL PTP4A3 PHOSPHATASE INHIBITORS UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2020-05-22 WO disclosed
WO-2020102245-A1 IN-FLOW PHOTOOXYGENATION OF AMINOTHIENOPYRIDINONES GENERATES NOVEL PTP4A3 PHOSPHATASE INHIBITORS UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2020-05-22 WO disclosed