SCHEMBL22017586

SCHEMBL22017586

Cc1ccc(NC(=O)c2ccc(OCCCCl)c([N+](=O)[O-])c2)cc1C(F)(F)F

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMPRSS2 O15393 1/20 0.57
POLB P06746 5/20 0.53
CTDSP1 Q9GZU7 1/20 0.53
MAPT P10636 10/20 0.50
MEN1 O00255 7/20 0.50
KMT2A Q03164 7/20 0.50
ALDH1A1 P00352 6/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
HTT P42858 1/20 0.49
LMNA P02545 3/20 0.48
CYP3A4 P08684 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C19 P33261 1/20 0.47
TDP1 Q9NUW8 2/20 0.47
TSHR P16473 1/20 0.47
NPC1 O15118 1/20 0.47
MAPK1 P28482 1/20 0.47
RAB9A P51151 1/20 0.47
ATM Q13315 1/20 0.47
GAA P10253 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28537925 0.91 TMPRSS2 (0.58) TMPRSS2POLBCTDSP1MAPTMEN1
SCHEMBL22017771 0.84 MAPT (0.47) MAPTMEN1KMT2AHTTLMNA
SCHEMBL22017401 0.82 TMPRSS2 (0.68) TMPRSS2POLBMAPTLMNA
SCHEMBL22017753 0.81 TMPRSS2 (0.87) TMPRSS2POLBMAPTMEN1KMT2A
SCHEMBL28547627 0.81 MAPT (0.55) POLBCTDSP1MAPTMEN1KMT2A
SCHEMBL22017242 0.81 TMPRSS2 (0.65) TMPRSS2MAPTMEN1KMT2AALDH1A1
SCHEMBL10092719 0.80 MAPT (0.59) POLBMAPTMEN1KMT2AALDH1A1
SCHEMBL22017757 0.80 TMPRSS2 (0.67) TMPRSS2POLBMAPTLMNA
SCHEMBL22017407 0.80 TMPRSS2 (0.66) TMPRSS2POLBMAPTLMNA
SCHEMBL22017408 0.79 TMPRSS2 (0.79) TMPRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109503518-B Substituted biaryl amide compound and preparation method and application thereof 中国医学科学院医药生物技术研究所 2021-03-30 CN disclosed
WO-2020098710-A1 SUBSTITUTED BIS-ARYL AMIDE COMPOUND AND PREPARATION METHOD AND APPLICATION THEREFOR 中国医学科学院医药生物技术研究所 2020-05-22 WO disclosed
CN-109503518-A A kind of substituted double aromatic radical amide compounds and its preparation method and application 中国医学科学院医药生物技术研究所 2019-03-22 CN disclosed