SCHEMBL22018536

SCHEMBL22018536

CCn1c(SCC(=O)Nc2cccc3ncn(C)c23)nnc1C1C=CSC1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.47
RORC P51449 1/20 0.47
ALDH1A1 P00352 4/20 0.42
POLB P06746 2/20 0.42
TSHR P16473 4/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
ALOX15 P16050 1/20 0.40
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.39
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22018535 0.80 CYP3A4 (0.48) CYP3A4RORCALDH1A1POLBTSHR
SCHEMBL15983300 0.79 ALDH1A1 (0.63) CYP3A4ALDH1A1POLBTSHRHTT
SCHEMBL13832095 0.78 MEN1 (0.65) CYP3A4ALDH1A1POLBTSHRMEN1
SCHEMBL13831179 0.76 KMT2A (0.51) CYP3A4ALDH1A1TSHRMEN1KMT2A
SCHEMBL22018798 0.76 CYP3A4 (0.42) CYP3A4RORCALDH1A1POLBTSHR
SCHEMBL13831297 0.76 NPSR1 (0.64) ALDH1A1POLBTSHRMEN1KMT2A
SCHEMBL15983380 0.76 MEN1 (0.53) CYP3A4ALDH1A1POLBTSHRMEN1
SCHEMBL13831879 0.75 POLB (0.63) ALDH1A1POLBTSHRMEN1KMT2A
SCHEMBL13831648 0.74 MAPK1 (0.60) ALDH1A1MEN1KMT2AMAPK1HTT
SCHEMBL22018538 0.74 SMN1; SMN2 (0.46) CYP3A4ALDH1A1POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3653054-A1 COMPOSITION FOR INHIBITION OF INSECT SENSING Vanderbilt University (US) 2020-05-20 EP disclosed
US-20160244756-A1 NOVEL FORMATS FOR ORGANIC COMPOUNDS FOR USE IN RNA INTERFERENCE NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH INC. 2016-08-25 US disclosed