SCHEMBL2202879

SCHEMBL2202879

O=S(=O)(O)c1cc(Nc2nc(Cl)nc(N3CCOCC3)n2)ccc1C=Cc1ccc(Nc2nc(Cl)nc(N3CCOCC3)n2)cc1S(=O)(=O)O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.53
TSHR P16473 1/20 0.53
PTGS2 P35354 4/20 0.52
TDP1 Q9NUW8 1/20 0.51
CA12 O43570 5/20 0.49
CA1 P00915 5/20 0.49
CA2 P00918 5/20 0.49
CA9 Q16790 5/20 0.49
MAPT P10636 2/20 0.48
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
LMNA P02545 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
ALOX15 P16050 1/20 0.46
MAPK1 P28482 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CREBBP Q92793 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14391125 1.00 SMN1; SMN2 (0.53) SMN1; SMN2TSHRPTGS2TDP1CA12
SCHEMBL11728864 0.99 PTGS2 (0.52) SMN1; SMN2TSHRPTGS2TDP1CA12
SCHEMBL2222266 0.99 PTGS2 (0.52) SMN1; SMN2TSHRPTGS2TDP1CA12
SCHEMBL3927919 0.99 PTGS2 (0.52) SMN1; SMN2TSHRPTGS2TDP1CA12
SCHEMBL14391122 0.94 CA12 (0.56) SMN1; SMN2TSHRPTGS2TDP1CA12
SCHEMBL2203214 0.93 CA12 (0.57) SMN1; SMN2TSHRPTGS2TDP1CA12
SCHEMBL2221311 0.92 CA12 (0.58) SMN1; SMN2TSHRPTGS2TDP1CA12
SCHEMBL17328820 0.90 HSD17B10 (0.48) SMN1; SMN2TSHRPTGS2TDP1CA12
SCHEMBL2220185 0.90 USP2 (0.47) SMN1; SMN2TSHRPTGS2TDP1CA12
SCHEMBL3927939 0.89 PTGS2 (0.52) SMN1; SMN2TSHRPTGS2TDP1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2716466-B1 THERMAL RECORDING MATERIAL CONTAINING STILBENE DISULPHONIC ACID FLUORESCENT WHITENING AGENT RICOH IND FRANCE SAS (FR) 2016-09-14 EP disclosed
EP-2722190-B1 Optimized undercoat for thermal recording material RICOH IND FRANCE SAS (FR) 2015-12-16 EP disclosed
EP-2722190-A1 Optimized undercoat for thermal recording material Ricoh Industrie France SAS (FR) 2014-04-23 EP disclosed
US-8546300-B2 Thermosensitive recording material and image recording method RICOH COMPANY, LTD. (JP) 2013-10-01 US disclosed
EP-2345541-B1 Thermosensitive recording material and image recording method RICOH CO LTD (JP) 2012-08-29 EP disclosed
US-20110177941-A1 THERMOSENSITIVE RECORDING MATERIAL AND IMAGE RECORDING METHOD RICOH COMPANY, LTD. (JP) 2011-07-21 US disclosed
EP-2345541-A2 Thermosensitive recording material and image recording method Ricoh Company, Ltd. (JP) 2011-07-20 EP disclosed
EP-1606380-B1 DETERGENT COMPOSITIONS CIBA SC HOLDING AG (CH) 2007-04-11 EP disclosed
EP-1485460-B1 PROCESS FOR THE TREATMENT OF TEXTILE FIBRE MATERIALS CIBA SC HOLDING AG (CH) 2006-09-27 EP disclosed
EP-1478724-B1 PROCESS FOR THE TREATMENT OF TEXTILE FIBRE MATERIALS CIBA SC HOLDING AG (CH) 2006-09-20 EP disclosed
EP-1606380-A1 DETERGENT COMPOSITIONS Ciba SC Holding AG (CH) 2005-12-21 EP disclosed
EP-1485460-A1 PROCESS FOR THE TREATMENT OF TEXTILE FIBRE MATERIALS Ciba SC Holding AG (CH) 2004-12-15 EP disclosed
EP-1478724-A1 PROCESS FOR THE TREATMENT OF TEXTILE FIBRE MATERIALS Ciba SC Holding AG (CH) 2004-11-24 EP disclosed
WO-2004085594-A1 DETERGENT COMPOSITIONS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2004-10-07 WO disclosed
WO-2003070869-A1 PROCESS FOR THE TREATMENT OF TEXTILE FIBRE MATERIALS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2003-08-28 WO disclosed
WO-2003070870-A1 PROCESS FOR THE TREATMENT OF TEXTILE FIBRE MATERIALS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2003-08-28 WO disclosed