SCHEMBL220296

SCHEMBL220296

CCCC(=O)ON1CCCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
L3MBTL1 Q9Y468 4/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CES2 O00748 1/20 0.35
CES1 P23141 1/20 0.35
RAB9A P51151 3/20 0.33
FFAR3 O14843 2/20 0.33
HDAC3 O15379 2/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC2 Q92769 2/20 0.33
HDAC8 Q9BY41 2/20 0.33
NPC1 O15118 2/20 0.33
TP53 P04637 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
SLC18A3 Q16572 1/20 0.33
ATM Q13315 1/20 0.32
TSHR P16473 1/20 0.32
MAPT P10636 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8433432 1.00 ALDH1A1 (0.46) ALDH1A1L3MBTL1MEN1KMT2ATDP1
SCHEMBL4124283 0.98 ALDH1A1 (0.44) ALDH1A1L3MBTL1MEN1KMT2ATDP1
SCHEMBL27474184 0.96 ALDH1A1 (0.43) ALDH1A1L3MBTL1MEN1KMT2ATDP1
Hydrochloric Acid SCHEMBL28611075 0.96 ALDH1A1 (0.43) ALDH1A1L3MBTL1MEN1KMT2ATDP1
SCHEMBL1535851 0.91
SCHEMBL28413576 0.88 L3MBTL1 (0.46) ALDH1A1L3MBTL1MEN1KMT2ATDP1
SCHEMBL8430106 0.86 L3MBTL1 (0.53) L3MBTL1MEN1KMT2ATDP1CES2
SCHEMBL5874880 0.86 L3MBTL1 (0.47) ALDH1A1L3MBTL1MEN1KMT2ATDP1
SCHEMBL8431983 0.84 L3MBTL1 (0.52) ALDH1A1L3MBTL1MEN1KMT2ATDP1
SCHEMBL8430031 0.84 L3MBTL1 (0.52) ALDH1A1L3MBTL1MEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 158 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080312267-A1 Diagnosis and Treatment of Diseases Arising from Defects in the Tuberous Sclerosis Pathway THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2008-12-18 US claimed
CN-100374158-C Diagnosis and treatment of the tuberous sclerosis pathway UNIV MICHIGAN (US) 2008-03-12 CN claimed
US-20250223297-A1 NOVEL RAPAMYCIN DERIVATIVES NOVARTIS AG (CH) 2025-07-10 US disclosed
CN-118804981-A Method for processing biomass material 普罗奥尼克股份有限公司 2024-10-18 CN disclosed
US-12091424-B2 Rapamycin derivatives NOVARTIS AG (CH) 2024-09-17 US disclosed
EP-4384493-A1 FERROPTOSIS MODULATORS, PREPARATIONS, AND USES THEREOF Sironax Ltd (KY) 2024-06-19 EP disclosed
US-20240180894-A1 METHODS OF TREATING MENTAL AND/OR MOOD DISORDERS USING 2-BROMO-LSD ALONE OR IN COMBINATION WITH A MTOR INHIBITOR BETTERLIFE PHARMA INC (CA) 2024-06-06 US disclosed
EP-4365179-A2 NOVEL RAPAMYCIN DERIVATIVES Novartis AG (CH) 2024-05-08 EP disclosed
CN-114477249-B Method for preparing high-purity magnesium hydroxide and calcium sulfate by adopting calcium carbide furnace purification ash 龙岩紫云化学科技有限公司 2024-01-30 CN disclosed
CN-117417351-A rapamycin derivatives 诺华股份有限公司 2024-01-19 CN disclosed
EP-3687999-B1 RAPAMYCIN DERIVATIVES NOVARTIS AG (CH) 2024-01-03 EP disclosed
US-5212155-A And cyclosporin, antibiotics CALNE ROY (GB) 1993-05-18 US disclosed
WO-1992017490-A1 PHOSPHORUS CONTAINING COMPOUNDS AS INHIBITORS OF RETROVIRUSES THE UPJOHN COMPANY (US) 1992-10-15 WO disclosed
CN-1016507-B Process for preparation of forskolin derivatives NIPPON KAYAKU KK (JP) 1992-05-06 CN disclosed
US-5100899-A METHODS OF INHIBITING TRANSPLANT REJECTION IN MAMMALS USING RAPAMYCIN AND DERIVATIVES AND PRODRUGS THEREOF CALNE ROY (GB) 1992-03-31 US disclosed
EP-0429436-A2 Prodrugs of rapamycin THE UNIVERSITY OF KANSAS (US) 1991-05-29 EP disclosed
EP-0401747-A2 Use of rapamycin and derivatives and prodrugs thereof in the manufacture of a medicament for inhibiting transplant rejection in mammals Calne, Roy (GB) 1990-12-12 EP disclosed
CN-86107826-A New forskrine derivant 1987-10-14 CN disclosed
EP-0227355-A2 Prodrugs of rapamycin THE UNIVERSITY OF KANSAS (US) 1987-07-01 EP disclosed
US-4650803-A WATER-SOLUBLE ANTITUMOR AGENTS UNIVERSITY OF KANSAS (US) 1987-03-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12091424-B2 Rapamycin derivatives RICTOR, MTOR, RPTOR ALDH1A1 3643/4885L3MBTL1 3400/4885MEN1 446/4885
US-20250223297-A1 NOVEL RAPAMYCIN DERIVATIVES MTOR, RICTOR, RPTOR ALDH1A1 4143/4885L3MBTL1 3265/4885MEN1 564/4885
US-20240180894-A1 METHODS OF TREATING MENTAL AND/OR MOOD DISORDERS USING 2-BROMO-LSD ALONE OR IN COMBINATION WITH A MTOR INHIBITOR MTOR, RICTOR, RPTOR ALDH1A1 4604/4885L3MBTL1 1489/4885MEN1 1710/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.