SCHEMBL22030682

SCHEMBL22030682

C=C1CCN(C(=O)CNC)Cc2c1c(=O)c(O)c1n2CCN(Cc2ccc(F)c(Cl)c2)C1=O

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CLPP Q16740 5/20 0.34
ENPP2 Q13822 1/20 0.33
KCNH2 Q12809 1/20 0.33
MAPK1 P28482 1/20 0.30
MAOB P27338 1/20 0.30
DPP4 P27487 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16185204 0.89 ENPP2 (0.34) CLPPENPP2KCNH2MAPK1DPP4
SCHEMBL16185213 0.86 CLPP (0.33) CLPPENPP2KCNH2MAPK1
SCHEMBL22030468 0.83 TP53 (0.34) CLPPENPP2KCNH2
SCHEMBL22030686 0.83 TP53 (0.34) CLPPENPP2KCNH2
SCHEMBL17547429 0.80 CLPP (0.35) CLPPKCNH2
SCHEMBL16185238 0.78 CLPP (0.34) CLPPKCNH2MAPK1
SCHEMBL16185260 0.76 ERCC1 (0.36) CLPPKCNH2MAPK1MAOB
SCHEMBL22031051 0.74 EGLN1 (0.35)
SCHEMBL16185211 0.74 CLPP (0.35) CLPPENPP2KCNH2
SCHEMBL16185205 0.73 ENPP2 (0.35) CLPPENPP2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2986291-B1 4-PYRIDONE DERIVATIVE COMPOUNDS AND USES THEREOF AS HIV INTEGRASE INHIBITORS MERCK SHARP & DOHME (US) 2020-05-27 EP disclosed