SCHEMBL22035587

SCHEMBL22035587

Cc1cc(-c2cn(CC3CC3)c(=O)c(C)n2)ccc1C#N

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 4/20 0.45
XDH P47989 2/20 0.40
GRM2 Q14416 5/20 0.40
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
BRD4 O60885 2/20 0.37
BAZ2A Q9UIF9 2/20 0.37
RPS6KB1 P23443 1/20 0.37
AKT1 P31749 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22031458 0.73 KDM1A (0.81) KDM1ARPS6KB1AKT1
SCHEMBL17375939 0.72 KDM1A (0.81) KDM1ARPS6KB1
SCHEMBL22035592 0.67 KDM1A (0.63) KDM1ACYP11B1CYP11B2
SCHEMBL13001686 0.63 TSHR (0.52) CYP11B1CYP11B2
SCHEMBL28918484 0.62 XDH (0.66) XDH
SCHEMBL16651145 0.60 BRD4 (0.40) GRM2BRD4BAZ2A
SCHEMBL22703631 0.60 BRD4 (0.54) BRD4BAZ2A
SCHEMBL19924644 0.59 BRD4 (0.65) BRD4BAZ2A
SCHEMBL18275112 0.59 AR (0.67)
SCHEMBL1816526 0.59 S1PR1 (0.41) CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3160956-B1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RES INC (US) 2020-05-27 EP disclosed