SCHEMBL2204502

SCHEMBL2204502

CCOC(=O)c1cc2c(Br)cccc2[nH]1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.55
ALDH1A1 P00352 5/20 0.55
RAB9A P51151 4/20 0.55
SMN1; SMN2 Q16637 4/20 0.55
MAPT P10636 4/20 0.55
HPGD P15428 3/20 0.55
NPC1 O15118 3/20 0.55
LMNA P02545 3/20 0.55
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
GLA P06280 1/20 0.55
GAA P10253 1/20 0.55
ATM Q13315 1/20 0.55
HSD17B10 Q99714 1/20 0.52
HRH4 Q9H3N8 1/20 0.52
HCRTR1 O43613 2/20 0.50
FLT3 P36888 1/20 0.50
ALOX15 P16050 1/20 0.50
HTT P42858 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL701020 0.85 KDM4E (0.57) KDM4EALDH1A1RAB9ASMN1; SMN2MAPT
SCHEMBL22620711 0.84 KDM4E (0.56) KDM4EALDH1A1RAB9ASMN1; SMN2MAPT
SCHEMBL913891 0.84 KDM4E (0.56) KDM4EALDH1A1RAB9ASMN1; SMN2MAPT
SCHEMBL2205092 0.84 HRH4 (0.56) KDM4EALDH1A1MAPTHPGDLMNA
SCHEMBL4044123 0.83 CDK1 (0.57) KDM4EALDH1A1RAB9ASMN1; SMN2MAPT
SCHEMBL5622391 0.83 KDM4E (0.55) KDM4EALDH1A1RAB9ASMN1; SMN2MAPT
SCHEMBL6303402 0.83 KDM4E (0.55) KDM4EALDH1A1RAB9ASMN1; SMN2MAPT
SCHEMBL5780732 0.83 KDM4E (0.56) KDM4EALDH1A1RAB9ASMN1; SMN2MAPT
SCHEMBL15904734 0.83 KDM4E (0.55) KDM4EALDH1A1RAB9ASMN1; SMN2MAPT
SCHEMBL25203298 0.82 KDM4E (0.56) KDM4EALDH1A1RAB9ASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 76 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113272276-A N-acyl sulfonamide salt FBPase inhibitor, preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2021-08-17 CN claimed
CN-111269167-A N-acyl sulfonamide salt FBPase inhibitor, preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2020-06-12 CN claimed
WO-2020114457-A1 N-ACYL SULFONAMIDE SALT FBPASE INHIBITOR, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION, AND USES THEREOF 中国医学科学院药物研究所 2020-06-11 WO claimed
EP-2948454-B1 TRIAZINE COMPOUNDS AND A PROCESS FOR PREPARATION THEREOF COUNCIL OF SCIENT & IND RES AN INDIAN REGISTERED BODY INCORPORATED UNDER THE REGISTRATION OF SOCIETI (IN) 2017-05-31 EP claimed
US-9447105-B2 Triazine compounds and a process for preparation thereof COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2016-09-20 US claimed
US-20150353566-A1 TRIAZINE COMPOUNDS AND A PROCESS FOR PREPARATION THEREOF COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2015-12-10 US claimed
EP-2948454-A1 TRIAZINE COMPOUNDS AND A PROCESS FOR PREPARATION THEREOF Council of Scientific & Industrial Research An Indian registered body incorporated under the Registration of Societies Act (Act XXI of 1860) (IN) 2015-12-02 EP claimed
WO-2014115171-A1 TRIAZINE COMPOUNDS AND A PROCESS FOR PREPARATION THEREOF COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2014-07-31 WO claimed
WO-2025067429-A1 COMPOUNDS, PREPARATION METHODS AND USES THEREOF InventisBio Co., Ltd. (CN) 2025-04-03 WO disclosed
US-20240043436-A1 METHODS AND COMPOUNDS FOR RESTORING MUTANT p53 FUNCTION PMV PHARMACEUTICALS, INC. 2024-02-08 US disclosed
WO-2023244672-A1 2-(IMIDAZO[1, 2-A]1,8-NAPHTHYRIDIN-8-YL)-1,3,4-OXADIAZOLE DERIVATIVES AS ENHANCERS OF INNATE IMMUNE RESPONSE FOR THE TREATMENT OF VIRAL INFECTIONS ASSEMBLY BIOSCIENCES, INC. (US) 2023-12-21 WO disclosed
US-11807644-B2 Methods and compounds for restoring mutant p53 function PMV PHARMACEUTICALS, INC. (US) 2023-11-07 US disclosed
US-11807644-B2 Methods and compounds for restoring mutant p53 function PMV PHARMACEUTICALS, INC. (US) 2023-11-07 US disclosed
EP-3962909-B1 NOVEL OXALYL PIPERAZINES ACTIVE AGAINST THE HEPATITIS B VIRUS (HBV) AICURIS GMBH & CO KG (DE) 2023-10-04 EP disclosed
US-6337344-B1 ANTICOAGULANTS AND ENZYME INHIBITORS FOR CARDIOVASCULAR DISORDERS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2002-01-08 US disclosed
WO-2001064639-A2 PDE IV INHIBITING AMIDES, COMPOSITIONS AND PHARMACEUTICAL USE MERCK FROSST CANADA & CO. (CA) 2001-09-07 WO disclosed
EP-1042287-A1 INDOLE DERIVATIVES AS INHIBITORS OF FACTOR XA Aventis Pharma Deutschland GmbH (DE) 2000-10-11 EP disclosed
EP-1003504-A2 INDOLE DERIVATIVES AND THEIR USE AS MCP-1 ANTAGONISTS AstraZeneca UK Limited (GB) 2000-05-31 EP disclosed
WO-1999033800-A1 INDOLE DERIVATIVES AS INHIBITORS OR FACTOR XA AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 1999-07-08 WO disclosed
WO-1999007351-A2 INDOLE DERIVATIVES AND THEIR USE AS MCP-1 ANTAGONISTS ZENECA LIMITED (GB) 1999-02-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150353566-A1 TRIAZINE COMPOUNDS AND A PROCESS FOR PREPARATION THEREOF TPH2, IDO2, INMT KDM4E 862/4885ALDH1A1 2885/4885RAB9A 4448/4885
US-11807644-B2 Methods and compounds for restoring mutant p53 function TP53, TP53BP1, HRAS KDM4E 3311/4885ALDH1A1 1977/4885RAB9A 1930/4885
US-20240043436-A1 METHODS AND COMPOUNDS FOR RESTORING MUTANT p53 FUNCTION TP53, TP53BP1, HRAS KDM4E 3311/4885ALDH1A1 1977/4885RAB9A 1930/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.