SCHEMBL22048060

SCHEMBL22048060

COC(=O)c1cnc(C2CCC(=O)CC2)s1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 1/20 0.41
HRH3 Q9Y5N1 2/20 0.38
HCRTR2 O43614 1/20 0.37
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
KMT2A Q03164 1/20 0.35
FFAR2 O15552 1/20 0.34
PARP1 P09874 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
MAPKAPK2 P49137 1/20 0.33
HPGD P15428 4/20 0.33
KDM4E B2RXH2 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
LMNA P02545 2/20 0.33
PPARG P37231 1/20 0.33
NCOA2 Q15596 1/20 0.33
NCOA1 Q15788 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22579415 0.90 HRH3 (0.41) CRBNHRH3HCRTR2ALDH1A1MEN1
SCHEMBL31704833 0.83 LRRK2 (0.40) CRBNHRH3HCRTR2ALDH1A1FFAR2
SCHEMBL14164278 0.83 HRH3 (0.38) CRBNHRH3HCRTR2ALDH1A1MEN1
SCHEMBL31706232 0.83 PLAT (0.41) CRBNHRH3HCRTR2MEN1KMT2A
SCHEMBL14164237 0.83 PLAT (0.41) CRBNHRH3HCRTR2MEN1KMT2A
SCHEMBL14164274 0.82 HRH3 (0.37) CRBNHRH3HCRTR2ALDH1A1MEN1
SCHEMBL14164234 0.82 HRH3 (0.42) CRBNHRH3HCRTR2SMN1; SMN2HTT
SCHEMBL628287 0.81 GSK3B (0.37) HRH3HCRTR2
SCHEMBL745563 0.75 GRM5 (0.43) CRBNALDH1A1HTTHPGDL3MBTL1
SCHEMBL14164236 0.75 GPR119 (0.48) CRBNHRH3ALDH1A1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020108579-A1 AMINO-SUBSTITUTED PYRIDONE DERIVATIVE, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL USE THEREOF 上海海雁医药科技有限公司 2020-06-04 WO disclosed