SCHEMBL2204873

SCHEMBL2204873

[c]1cncn1C(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 3/20 0.44
CYP11B2 P19099 3/20 0.44
KCNN4 O15554 3/20 0.36
TSHR P16473 3/20 0.36
NR1I2 O75469 2/20 0.36
ADORA3 P0DMS8 2/20 0.36
TBXA2R P21731 2/20 0.36
CCKBR P32239 2/20 0.36
OPRK1 P41145 2/20 0.36
SLC6A3 Q01959 2/20 0.36
KCNH2 Q12809 2/20 0.36
NR1H4 Q96RI1 2/20 0.36
KCNA3 P22001 2/20 0.36
CYP3A4 P08684 2/20 0.36
MEN1 O00255 1/20 0.36
SLC22A1 O15245 1/20 0.36
GMNN O75496 1/20 0.36
USP2 O75604 1/20 0.36
TRPM2 O94759 1/20 0.36
ABCB11 O95342 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1292257 0.64 CYP11B1 (0.44) CYP11B1CYP11B2KCNN4TSHRNR1I2
SCHEMBL4800641 0.64 CYP3A4 (0.39) TSHRCYP3A4MEN1EGFRALOX15
SCHEMBL30577371 0.63 CYP11B1 (0.57) CYP11B1CYP11B2KCNN4TSHRNR1I2
SCHEMBL332630 0.61 CYP11B1 (1.00) CYP11B1CYP11B2KCNN4TSHRNR1I2
SCHEMBL9602007 0.61 KCNN4 (0.38) CYP11B1CYP11B2KCNN4TSHRNR1I2
SCHEMBL1563373 0.61 HSP90AA1 (0.47) CYP11B1CYP11B2KCNN4TSHRNR1I2
SCHEMBL2204870 0.60 CYP11B1 (0.48) CYP11B1CYP11B2KCNN4TSHRNR1I2
SCHEMBL8443367 0.60 CYP11B1 (0.40) CYP11B1CYP11B2KCNN4TSHRNR1I2
SCHEMBL8443085 0.60 CYP11B1 (0.36) CYP11B1CYP11B2KCNN4TSHRKCNA3
SCHEMBL1757361 0.60 CYP11B1 (0.40) CYP11B1CYP11B2KCNN4TSHRNR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101711242-B ((bicyclic heteroaryl) imidazolyl) methyl heteroaryl compounds as adrenergic receptor agonists ALLERGAN INC 2013-09-25 CN disclosed
CN-101743240-B ((phenyl) imidazolyl) methyl heteroaryl compounds ALLERGAN INC 2013-07-17 CN disclosed
EP-2079706-B1 METHOD FOR PREPARING MEDETOMIDINE AND ITS SALTS GRINDEKS JSC (LV) 2011-07-20 EP disclosed
CN-101743240-A ((phenyl) imidazolyl) methyl heteroaryl compounds ALLERGAN INC 2010-06-16 CN disclosed
CN-101711242-A ((bicyclic heteroaryl) imidazolyl) methyl heteroaryl compounds as adrenergic receptor agonists ALLERGAN INC 2010-05-19 CN disclosed
US-5643878-A TREATMENT OF RETROVIRAL DISEASES LIKE AIDS CIBA-GEIGY CORPORATION (US) 1997-07-01 US disclosed
EP-0618222-A2 Dipeptid derivatives of 5-amino-4-hydroxy-hexanoic acid CIBA-GEIGY AG (CH) 1994-10-05 EP disclosed