SCHEMBL8443085

SCHEMBL8443085

[c]1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)nn1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
KCNN4 O15554 2/20 0.33
KCNA3 P22001 1/20 0.33
TSHR P16473 2/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9602007 0.69 KCNN4 (0.38) CYP11B1CYP11B2KCNN4KCNA3TSHR
SCHEMBL7982989 0.68 CYP11B1 (0.40) CYP11B1CYP11B2KCNN4KCNA3TSHR
SCHEMBL1563373 0.65 HSP90AA1 (0.47) CYP11B1CYP11B2KCNN4KCNA3TSHR
SCHEMBL1197948 0.65 CYP11B1 (0.37) CYP11B1CYP11B2KCNN4KCNA3TSHR
SCHEMBL198143 0.65 NOTUM (0.45) CYP11B1CYP11B2KCNN4KCNA3TSHR
SCHEMBL7796676 0.65 CYP11B1 (0.46) CYP11B1CYP11B2KCNN4KCNA3TSHR
SCHEMBL2204870 0.64 CYP11B1 (0.48) CYP11B1CYP11B2KCNN4KCNA3TSHR
SCHEMBL8443367 0.64 CYP11B1 (0.40) CYP11B1CYP11B2KCNN4KCNA3TSHR
SCHEMBL2036810 0.64 CYP11B1 (0.36) CYP11B1CYP11B2KCNN4KCNA3TSHR
SCHEMBL2392374 0.63 KCNN4 (0.69) CYP11B1CYP11B2KCNN4KCNA3TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0594263-B1 INTERMEDIATES FOR THE PREPARATION OF THIOALKYLTHIO CEPHALOSPORIN DERIVATIVES SHIONOGI & CO (JP) 1999-06-09 EP disclosed
CN-1034504-C Thioalkylthio cephalosporin derivatives SHIONOGI & CO (JP) 1997-04-09 CN disclosed
US-5352792-A Bactericides SHIONOGI & CO., LTD. (JP) 1994-10-04 US disclosed
EP-0467647-B1 Thioalkylthio cephalosporin derivatives SHIONOGI & CO (JP) 1994-08-17 EP disclosed
EP-0594263-A1 Thioalkylthio cephalosporin derivatives and intermediates SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1994-04-27 EP disclosed
US-5214037-A Antibiotic, bactericide SHIONOGI & CO., LTD. (JP) 1993-05-25 US disclosed
EP-0467647-A2 Thioalkylthio cephalosporin derivatives SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1992-01-22 EP disclosed