SCHEMBL22061332

SCHEMBL22061332

COC(=O)c1ccc(C(=O)C(C)C)nc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.72
KDM4E B2RXH2 2/20 0.68
L3MBTL1 Q9Y468 1/20 0.68
ALDH1A1 P00352 3/20 0.45
PLA2G1B P04054 1/20 0.43
ATG4B Q9Y4P1 1/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
CA12 O43570 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
KMT2A Q03164 3/20 0.43
RAB9A P51151 2/20 0.43
NPC1 O15118 1/20 0.43
P4HTM Q9NXG6 3/20 0.42
MAPT P10636 2/20 0.42
P4HA1 P13674 1/20 0.42
MIF P14174 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10060485 0.86 P4HTM (0.50) MAPK1KDM4EL3MBTL1ALDH1A1KMT2A
SCHEMBL69747 0.84 MAPK1 (1.00) MAPK1KDM4EL3MBTL1ALDH1A1CA1
SCHEMBL29508473 0.84 MAPK1 (1.00) MAPK1KDM4EL3MBTL1ALDH1A1CA1
SCHEMBL1018248 0.82 MAPK1 (0.70) MAPK1KDM4EL3MBTL1ALDH1A1PLA2G1B
SCHEMBL64700 0.81 MAPK1 (1.00) MAPK1KDM4EL3MBTL1P4HTMP4HA1
SCHEMBL423045 0.81 MAPK1 (0.79) MAPK1KDM4EL3MBTL1ALDH1A1CA1
SCHEMBL16185858 0.81 P4HTM (0.46) MAPK1KDM4EL3MBTL1ALDH1A1KMT2A
SCHEMBL22060647 0.81 P4HTM (0.66) MAPK1KDM4EL3MBTL1ALDH1A1P4HTM
SCHEMBL4295029 0.80 MAPK1 (0.62) MAPK1KDM4EL3MBTL1ALDH1A1PLA2G1B
SCHEMBL2656944 0.80 CA1 (0.59) KDM4EL3MBTL1ALDH1A1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020108538-A1 RORγ INHIBITOR HAVING SULFONYL STRUCTURE 正大天晴药业集团股份有限公司 2020-06-04 WO disclosed