SCHEMBL22064465

SCHEMBL22064465

C=CCC1(F)CN(C(=O)OC(C)(C)C)CCC1Oc1cc(C#N)c(/N=C\N(C)C)cc1OC

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 7/20 0.35
NSD2 O96028 2/20 0.35
PDE4B Q07343 5/20 0.35
PDE4A P27815 4/20 0.35
PDE4C Q08493 4/20 0.35
PDE4D Q08499 4/20 0.35
EHMT2 Q96KQ7 2/20 0.33
KDM1A O60341 1/20 0.33
RCOR1 Q9UKL0 1/20 0.33
IKBKE Q14164 2/20 0.33
TBK1 Q9UHD2 2/20 0.33
EGFR P00533 1/20 0.32
PIK3CD O00329 2/20 0.31
PIK3CA P42336 2/20 0.31
PIK3CB P42338 2/20 0.31
PIK3CG P48736 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20709081 0.89 GPR119 (0.38) GPR119NSD2PDE4BPDE4APDE4C
SCHEMBL30727149 0.89 GPR119 (0.38) GPR119NSD2PDE4BPDE4APDE4C
SCHEMBL28405729 0.89 GPR119 (0.38) GPR119NSD2PDE4BPDE4APDE4C
SCHEMBL22064466 0.87 GPR119 (0.37) GPR119NSD2PDE4BPDE4APDE4C
SCHEMBL5048849 0.79 GPR119 (0.42) GPR119NSD2PDE4BPDE4APDE4C
SCHEMBL5048852 0.79 GPR119 (0.42) GPR119NSD2PDE4BPDE4APDE4C
SCHEMBL21473543 0.75 STS (0.37) GPR119NSD2PDE4BPDE4APDE4C
SCHEMBL21481104 0.74 TBK1 (0.36) NSD2TBK1EGFR
SCHEMBL30126189 0.74 NSD2 (0.35) GPR119NSD2PDE4BEHMT2PIK3CD
SCHEMBL30125949 0.74 NSD2 (0.35) GPR119NSD2PDE4BEHMT2PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3438107-B1 SUBSTITUTED QUINAZOLINE COMPOUND HAVING BLOOD-BRAIN BARRIER PENETRATION CAPABILITY WEISHANG SHANGHAI BIO PHARMACEUTICAL CO LTD (CN) 2020-06-10 EP disclosed