SCHEMBL22065286

SCHEMBL22065286

CNc1cc(C(=O)Nc2cccc(F)c2)ccc1C

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRAF P15056 3/20 0.60
KCNK3 O14649 2/20 0.59
KCNK9 Q9NPC2 1/20 0.59
NPC1 O15118 5/20 0.58
RAB9A P51151 5/20 0.58
HPGD P15428 2/20 0.58
MEN1 O00255 6/20 0.56
KMT2A Q03164 6/20 0.56
CNR1 P21554 1/20 0.56
TSHR P16473 1/20 0.55
MAOB P27338 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
LCK P06239 1/20 0.51
KIT P10721 1/20 0.51
SRC P12931 1/20 0.51
MAPK14 Q16539 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22065295 0.88 KCNK3 (0.58) BRAFKCNK3KCNK9NPC1RAB9A
SCHEMBL22065291 0.86 MEN1 (0.68) KCNK3KCNK9NPC1RAB9AMEN1
SCHEMBL20922103 0.86 KCNK3 (0.65) BRAFKCNK3KCNK9NPC1RAB9A
SCHEMBL22024522 0.86 CNR1 (0.55) BRAFKCNK3KCNK9NPC1RAB9A
SCHEMBL22025348 0.86 CNR1 (0.55) BRAFKCNK3KCNK9NPC1RAB9A
SCHEMBL22065285 0.84 BRAF (0.60) BRAFKCNK3KCNK9NPC1RAB9A
SCHEMBL17131157 0.83 MAPK14 (0.72) BRAFKCNK3KCNK9RAB9AMEN1
SCHEMBL22025010 0.82 KCNK3 (0.60) BRAFKCNK3KCNK9NPC1RAB9A
SCHEMBL22066261 0.82 MAPK14 (0.64) BRAFKCNK3HPGDSMN1; SMN2MAPK14
SCHEMBL22065404 0.82 RXFP1 (0.68) KCNK3KCNK9NPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3663293-A1 SUBSTITUTED PENTA- AND HEXA-HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, DRUG COMBINATION AND USE THEREOF Xiamen University (CN) 2020-06-10 EP disclosed