SCHEMBL22069593

SCHEMBL22069593

CC(C)c1ccc(Oc2ccc([N+](=O)[O-])cc2Cl)cc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE7A Q13946 1/20 0.74
KMT2A Q03164 7/20 0.63
MEN1 O00255 6/20 0.63
GAA P10253 1/20 0.63
PKM P14618 1/20 0.63
ALDH1A1 P00352 7/20 0.59
MAPT P10636 7/20 0.56
KDM4E B2RXH2 1/20 0.55
LMNA P02545 3/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
HSPB1 P04792 2/20 0.49
HSD17B10 Q99714 1/20 0.47
GPR55 Q9Y2T6 1/20 0.46
HPGD P15428 2/20 0.46
NPC1 O15118 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22966266 0.86 PDE7A (0.55) PDE7AKMT2AMEN1GAAPKM
SCHEMBL11760667 0.85 PDE7A (1.00) PDE7AKMT2AMEN1GAAPKM
SCHEMBL2967458 0.85 PDE7A (0.78) PDE7AKMT2AMEN1GAAPKM
SCHEMBL22069751 0.84 HSPB1 (0.63) PDE7AKMT2AMEN1GAAPKM
SCHEMBL11198374 0.84 PDE7A (0.76) PDE7AKMT2AMEN1GAAPKM
SCHEMBL11195566 0.83 PDE7A (0.62) PDE7AKMT2AMEN1GAAPKM
SCHEMBL22069562 0.82 PDE7A (0.74) PDE7AKMT2AMEN1GAAPKM
SCHEMBL9367473 0.82 PDE7A (0.74) PDE7AKMT2AMEN1GAAPKM
SCHEMBL4029870 0.82 PDE7A (0.73) PDE7AKMT2AMEN1GAAPKM
SCHEMBL10856843 0.82 MEN1 (0.62) PDE7AKMT2AMEN1GAAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666769-A1 NOVEL CASPASE INHIBITORS RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-06-17 EP disclosed
EP-3666769-A1 NOVEL CASPASE INHIBITORS RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-06-17 EP disclosed