SCHEMBL22069596

SCHEMBL22069596

O=[N+]([O-])c1ccc(Oc2cccc(Cl)c2)c(F)c1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSPB1 P04792 6/20 0.56
EPAS1 Q99814 1/20 0.55
MEN1 O00255 5/20 0.53
KMT2A Q03164 5/20 0.53
ALDH1A1 P00352 5/20 0.53
MAPT P10636 4/20 0.53
LMNA P02545 3/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
TBXA2R P21731 2/20 0.53
TDP1 Q9NUW8 1/20 0.53
PDE7A Q13946 1/20 0.47
GPR55 Q9Y2T6 1/20 0.46
EYA2 O00167 1/20 0.44
HTT P42858 1/20 0.44
HIF1A Q16665 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28317228 0.89 ALDH1A1 (0.53) HSPB1EPAS1MEN1KMT2AALDH1A1
SCHEMBL22069742 0.87 HSPB1 (0.60) HSPB1EPAS1MEN1KMT2AALDH1A1
SCHEMBL2529627 0.86 ALDH1A1 (0.67) EPAS1MEN1KMT2AALDH1A1MAPT
SCHEMBL3845633 0.84 MEN1 (0.67) HSPB1EPAS1MEN1KMT2AALDH1A1
SCHEMBL22069708 0.84 HSPB1 (0.68) HSPB1MEN1KMT2AALDH1A1MAPT
SCHEMBL4082910 0.84 HSPB1 (0.68) HSPB1MEN1KMT2AALDH1A1MAPT
SCHEMBL124556 0.82 TBXA2R (0.54) EPAS1MEN1KMT2AALDH1A1MAPT
SCHEMBL22069594 0.82 HSPB1 (0.61) HSPB1EPAS1MEN1KMT2AALDH1A1
SCHEMBL14965155 0.81 HSPB1 (0.73) HSPB1MEN1KMT2AALDH1A1MAPT
SCHEMBL2035696 0.81 HSPB1 (0.53) HSPB1MEN1KMT2AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666769-A1 NOVEL CASPASE INHIBITORS RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-06-17 EP disclosed
EP-3666769-A1 NOVEL CASPASE INHIBITORS RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-06-17 EP disclosed