SCHEMBL22076876

SCHEMBL22076876

CN(C)C=Nc1ccc(NC(=O)COP(=O)(O)O)cc1C#N

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
KMT2A Q03164 3/20 0.36
TDP1 Q9NUW8 1/20 0.36
ALDH1A1 P00352 6/20 0.36
NAMPT P43490 1/20 0.35
GAA P10253 3/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35
S1PR1 P21453 1/20 0.35
S1PR3 Q99500 1/20 0.35
LMNA P02545 5/20 0.35
MEN1 O00255 1/20 0.35
HTT P42858 1/20 0.35
KCNH2 Q12809 1/20 0.34
HCRTR1 O43613 1/20 0.34
USP2 O75604 1/20 0.34
HPGD P15428 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22076875 1.00 NPC1 (0.37) NPC1RAB9AKMT2ATDP1ALDH1A1
SCHEMBL29025878 0.89 ALDH1A1 (0.38) NPC1RAB9AKMT2ATDP1ALDH1A1
SCHEMBL30478696 0.89 ALDH1A1 (0.38) NPC1RAB9AKMT2ATDP1ALDH1A1
SCHEMBL29025875 0.82 S1PR1 (0.40) ALDH1A1S1PR1S1PR3
SCHEMBL20605293 0.80 ALDH1A1 (0.40) NPC1RAB9AKMT2AALDH1A1GAA
SCHEMBL20605289 0.80 ALDH1A1 (0.40) NPC1RAB9AKMT2AALDH1A1GAA
SCHEMBL2249224 0.78 ALDH1A1 (0.37) KMT2ATDP1ALDH1A1GAALMNA
SCHEMBL19322331 0.77 ALDH1A1 (0.38) NPC1RAB9AKMT2AALDH1A1GAA
SCHEMBL24167727 0.76 EGFR (0.40) NPC1RAB9AKMT2AALDH1A1GAA
SCHEMBL6584471 0.76 EGFR (0.40) NPC1RAB9AKMT2AALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109422755-B Nitrogen-containing heterocyclic compound, preparation method, intermediate, composition and application 上海医药集团股份有限公司 2023-07-04 CN disclosed
US-11578074-B2 Nitrogenous heterocyclic compound, preparation method, intermediate, composition, and application Shanghai Pharmaceuticals Holding Cd., Ltd. (CN) 2023-02-14 US disclosed
EP-3677583-A1 NITROGENOUS HETEROCYCLIC COMPOUND, PREPARATION METHOD, INTERMEDIATE, COMPOSITION, AND APPLICATION Shanghai Pharmaceuticals Holding Co., Ltd. (CN) 2020-07-08 EP disclosed
US-20200190091-A1 NITROGENOUS HETEROCYCLIC COMPOUND, PREPARATION METHOD, INTERMEDIATE, COMPOSITION, AND APPLICATION SHANGHAI PHARMACEUTICALS HOLDING CO., LTD. (CN) 2020-06-18 US disclosed
CN-109422755-A A kind of nitrogen-containing heterocycle compound, preparation method, intermediate, composition and application 上海医药集团股份有限公司 2019-03-05 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200190091-A1 NITROGENOUS HETEROCYCLIC COMPOUND, PREPARATION METHOD, INTERMEDIATE, COMPOSITION, AND APPLICATION ERBB2, EGFR, ERBB4 NPC1 1519/4885RAB9A 1981/4885KMT2A 2737/4885
US-11578074-B2 Nitrogenous heterocyclic compound, preparation method, intermediate, composition, and application ERBB2, EGFR, ERBB4 NPC1 1553/4885RAB9A 2006/4885KMT2A 2632/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.