SCHEMBL22100012

SCHEMBL22100012

NCCOCCOCCNC(=O)c1cccc2c(N)ccc(C=O)c12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 2/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
KDM4E B2RXH2 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
MAPK1 P28482 2/20 0.36
TP53 P04637 1/20 0.36
HSD17B10 Q99714 1/20 0.36
HDAC3 O15379 2/20 0.34
HDAC1 Q13547 2/20 0.34
NQO2 P16083 1/20 0.34
CA2 P00918 2/20 0.33
PRKCD Q05655 2/20 0.33
CAMK2B Q13554 2/20 0.33
CAMK2G Q13555 2/20 0.33
AURKB Q96GD4 2/20 0.33
DAPK3 O43293 1/20 0.33
PRKD3 O94806 1/20 0.33
MAP4K4 O95819 1/20 0.33
CHEK2 O96017 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22099932 0.84 KDM4E (0.35) ALDH1A1HPGDKDM4ESMN1; SMN2TP53
SCHEMBL22100116 0.76 KDM4E (0.34) ALDH1A1HPGDKDM4ESMN1; SMN2HDAC3
SCHEMBL3486549 0.71 ALDH1A1 (0.41) NSD2ALDH1A1HPGDKDM4ESMN1; SMN2
SCHEMBL13692597 0.71 KDM4E (0.39) ALDH1A1HPGDKDM4ESMN1; SMN2CA2
SCHEMBL12708259 0.71 MEN1 (0.56) ALDH1A1HPGDKDM4ESMN1; SMN2MAPK1
SCHEMBL1584943 0.69 MEN1 (0.57) ALDH1A1HPGDKDM4ESMN1; SMN2MAPK1
SCHEMBL14669007 0.69 SMN1; SMN2 (0.51) ALDH1A1HPGDSMN1; SMN2MAPK1TP53
SCHEMBL16549869 0.69 SMN1; SMN2 (0.48) ALDH1A1HPGDSMN1; SMN2MAPK1TP53
SCHEMBL22124710 0.68 NPC1 (0.58) ALDH1A1HPGDSMN1; SMN2MAPK1TP53
SCHEMBL16329591 0.68 SMN1; SMN2 (0.50) ALDH1A1HPGDSMN1; SMN2MAPK1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2976081-B1 METHODS OF ACUTE RESTORATION OF VASCULAR COMPLIANCE ALUMEND LLC (US) 2020-06-17 EP disclosed