SCHEMBL22101280

SCHEMBL22101280

CCC(=O)c1ccc(Nc2cccnc2Nc2ccc(C#N)c(C(F)(F)F)c2)cc1F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS2R14 Q9NYV8 1/20 0.52
AR P10275 9/20 0.43
KDR P35968 2/20 0.41
BRAF P15056 1/20 0.41
TRPV1 Q8NER1 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
TUBB4A P04350 1/20 0.39
TUBB P07437 1/20 0.39
TUBA3C P0DPH7 1/20 0.39
TUBA1B P68363 1/20 0.39
TUBA4A P68366 1/20 0.39
TUBB4B P68371 1/20 0.39
TUBB3 Q13509 1/20 0.39
TUBB2A Q13885 1/20 0.39
TUBB8 Q3ZCM7 1/20 0.39
TUBA3E Q6PEY2 1/20 0.39
TUBA1A Q71U36 1/20 0.39
TUBA1C Q9BQE3 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22101261 0.89 TAS2R14 (0.54) TAS2R14ARKDRBRAFTRPV1
SCHEMBL22393602 0.74 TAS2R14 (0.44) TAS2R14ARKDRBRAFTRPV1
SCHEMBL20852437 0.69 AR (0.62) AR
SCHEMBL15131415 0.67 AR (0.54) ARCYP2D6CYP2C9CYP2C19
SCHEMBL18049814 0.67 KDR (0.63) ARKDR
SCHEMBL14916193 0.67 AR (0.55) ARKDRBRAF
SCHEMBL13653030 0.66 LMNA (0.74) ARCYP2D6CYP2C9CYP2C19
SCHEMBL22563041 0.66 TAS2R14 (0.56) TAS2R14AR
SCHEMBL9369888 0.65 AR (0.60) ARCYP2C19
SCHEMBL16946786 0.65 AR (0.54) AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666772-A1 DIARYLTHIOHYDANTOIN COMPOUND AS ANDROGEN RECEPTOR ANTAGONIST Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2020-06-17 EP disclosed