SCHEMBL22101448

SCHEMBL22101448

CCc1nc(CC)c2cc(Nc3c(C)ccnc3Nc3ccc(C#N)c(C(F)(F)F)c3)cc(F)c2n1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.39
ERBB2 P04626 1/20 0.38
TDO2 P48775 3/20 0.38
ABCG2 Q9UNQ0 1/20 0.37
MAP3K8 P41279 5/20 0.35
KDR P35968 3/20 0.35
AR P10275 3/20 0.34
NTSR1 P30989 1/20 0.34
VCP P55072 1/20 0.34
BRAF P15056 1/20 0.34
STK17A Q9UEE5 1/20 0.33
RORC P51449 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22101389 0.91 EGFR (0.41) EGFRERBB2TDO2ABCG2MAP3K8
SCHEMBL22101890 0.81 ABCG2 (0.41) EGFRERBB2TDO2ABCG2KDR
SCHEMBL22101880 0.76 AR (0.41) EGFRERBB2ABCG2MAP3K8AR
SCHEMBL22393602 0.75 TAS2R14 (0.44) EGFRERBB2KDRARBRAF
SCHEMBL22393849 0.75 ABCG2 (0.35) EGFRABCG2KDRARNTSR1
SCHEMBL22101394 0.65 BRAF (0.33) TDO2BRAF
SCHEMBL22101280 0.63 TAS2R14 (0.52) KDRARBRAF
SCHEMBL3938525 0.62 TRPV1 (0.68)
SCHEMBL3289311 0.59 AR (0.52) AR
SCHEMBL3057215 0.58 AR (0.55) AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666772-A1 DIARYLTHIOHYDANTOIN COMPOUND AS ANDROGEN RECEPTOR ANTAGONIST Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2020-06-17 EP disclosed