SCHEMBL22101758

SCHEMBL22101758

O=c1[nH]c(C2CC2)nc2c(F)cc(Br)cc12

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 8/20 0.47
PIM1 P11309 8/20 0.47
CSNK2B P67870 8/20 0.47
CSNK2A1 P68400 8/20 0.47
TMIGD3 P0DMS9 1/20 0.43
ADORA1 P30542 1/20 0.43
TNKS O95271 3/20 0.40
TNKS2 Q9H2K2 3/20 0.40
ROCK2 O75116 2/20 0.40
PARP1 P09874 1/20 0.38
TYK2 P29597 1/20 0.37
PARG Q86W56 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29800642 0.87 PARP1 (0.43) CDC7PIM1CSNK2BCSNK2A1TMIGD3
SCHEMBL27242013 0.87 PARP1 (0.43) CDC7PIM1CSNK2BCSNK2A1TMIGD3
SCHEMBL23293951 0.79 KDM4E (0.47)
SCHEMBL22101466 0.75 PARP1 (0.37) PIM1CSNK2BTNKSTNKS2PARP1
SCHEMBL25795251 0.73 CDC7 (0.38) CDC7PIM1CSNK2BCSNK2A1TMIGD3
SCHEMBL30783587 0.73 CDC7 (0.40) CDC7PIM1CSNK2BCSNK2A1TMIGD3
SCHEMBL22101792 0.73 PIM1 (0.38) CDC7PIM1CSNK2BCSNK2A1TNKS
SCHEMBL22393820 0.73 PKM (0.46) PIM1CSNK2BCSNK2A1TNKSTNKS2
SCHEMBL22600708 0.72 CDC7 (0.37) CDC7PIM1CSNK2BCSNK2A1TMIGD3
SCHEMBL22101365 0.72 PARP1 (0.47) PIM1CSNK2BADORA1TNKSTNKS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666772-A1 DIARYLTHIOHYDANTOIN COMPOUND AS ANDROGEN RECEPTOR ANTAGONIST Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2020-06-17 EP disclosed