SCHEMBL22101759

SCHEMBL22101759

CCc1nc(=O)c2cc(Br)cc(C)c2[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 5/20 0.46
PARP4 Q9UKK3 2/20 0.39
PARP1 P09874 1/20 0.39
PARP2 Q9UGN5 1/20 0.39
ADORA3 P0DMS8 4/20 0.36
ADORA2A P29274 3/20 0.36
TNKS2 Q9H2K2 1/20 0.36
GSK3B P49841 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.33
TP53 P04637 1/20 0.33
TYMS P04818 1/20 0.32
KMT2A Q03164 1/20 0.32
GAA P10253 2/20 0.31
NLRP3 Q96P20 1/20 0.31
HTT P42858 1/20 0.31
ALDH1A1 P00352 2/20 0.31
KDM4E B2RXH2 1/20 0.31
CACNA1B Q00975 1/20 0.31
APBA1 Q02410 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22393745 0.84 ADORA1 (0.36) ADORA1PARP4PARP1PARP2ADORA3
SCHEMBL1918902 0.78 ADORA1 (0.51) ADORA1PARP4PARP1PARP2ADORA3
SCHEMBL22101275 0.76 PARP4 (0.63) PARP4PARP1PARP2TNKS2L3MBTL1
SCHEMBL22101352 0.74 PRNP (0.48) TNKS2GSK3BSMN1; SMN2TYMSKMT2A
SCHEMBL22101768 0.69 PIM1 (0.41) PARP4PARP1PARP2GSK3BKMT2A
SCHEMBL1128687 0.68 NQO2 (0.47) TNKS2GSK3BSMN1; SMN2TP53GAA
SCHEMBL1918900 0.68 EGLN1 (0.42) ADORA1PARP4PARP1PARP2ADORA3
SCHEMBL3210466 0.68 ADORA1 (0.70) ADORA1ADORA3ADORA2ASMN1; SMN2L3MBTL1
SCHEMBL3208633 0.68 GSK3B (0.38) PARP4PARP1PARP2GSK3B
SCHEMBL16167174 0.67 GSK3B (0.39) PARP4PARP1PARP2GSK3BSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666772-A1 DIARYLTHIOHYDANTOIN COMPOUND AS ANDROGEN RECEPTOR ANTAGONIST Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2020-06-17 EP disclosed