SCHEMBL22101768

SCHEMBL22101768

Cc1cc(Br)cc2c(=O)nc[nH]c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 3/20 0.41
PIM3 Q86V86 2/20 0.41
CHEK1 O14757 2/20 0.41
AKT1 P31749 1/20 0.41
FLT3 P36888 1/20 0.41
PARP1 P09874 5/20 0.38
ALDH1A1 P00352 1/20 0.35
PDPK1 O15530 1/20 0.35
CSNK2A2 P19784 2/20 0.35
CSNK2B P67870 2/20 0.35
CSNK2A1 P68400 2/20 0.35
CSNK2A3 Q8NEV1 2/20 0.35
CDC7 O00311 1/20 0.35
PIM2 Q9P1W9 1/20 0.35
PARP2 Q9UGN5 1/20 0.35
PARP4 Q9UKK3 1/20 0.35
RPS6KA3 P51812 1/20 0.34
MEN1 O00255 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3226647 0.79 PIM1 (0.41) PIM1PIM3CHEK1AKT1FLT3
SCHEMBL2418830 0.76 NQO2 (0.38) PIM1PIM3CHEK1AKT1FLT3
SCHEMBL31056362 0.76 NQO2 (0.38) PIM1PIM3CHEK1AKT1FLT3
SCHEMBL20680534 0.75 PARP1 (0.39) PIM1PIM3CHEK1AKT1FLT3
SCHEMBL16112933 0.74 PARP1 (0.70) PIM1PIM3CHEK1AKT1FLT3
SCHEMBL5370069 0.73 PARP1 (0.54) CHEK1PARP1PDPK1
SCHEMBL22492390 0.71 CCR8 (0.48) PIM3ALDH1A1KMT2AHPGD
SCHEMBL1144808 0.71 GSK3B (0.36) GSK3B
SCHEMBL17030854 0.70 PARP1 (0.37) PIM1CHEK1PARP1ALDH1A1PDPK1
SCHEMBL22101759 0.69 ADORA1 (0.46) PARP1ALDH1A1PARP2PARP4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666772-A1 DIARYLTHIOHYDANTOIN COMPOUND AS ANDROGEN RECEPTOR ANTAGONIST Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2020-06-17 EP disclosed