SCHEMBL22112248

SCHEMBL22112248

Oc1cc(F)c(F)c(C[C@H]2CC=C(c3ccccc3)CC2)c1

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.45
CYP26A1 O43174 1/20 0.33
DRD2 P14416 2/20 0.32
DRD3 P35462 2/20 0.32
DRD4 P21917 1/20 0.32
HRH3 Q9Y5N1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22112044 0.88 ESR2 (0.43) ESR2CYP26A1DRD2DRD3DRD4
SCHEMBL22112048 0.74 ESR2 (0.49) ESR2DRD2DRD3
SCHEMBL22112254 0.69 ESR2 (0.44) ESR2
SCHEMBL22112200 0.68 RIPK1 (0.31)
SCHEMBL10931209 0.67 ESR2 (0.49) ESR2DRD2DRD3DRD4
SCHEMBL10091140 0.66 ESR2 (0.38) ESR2
SCHEMBL22112337 0.66 ALDH1A1 (0.42) ESR2DRD2DRD3DRD4
SCHEMBL10931202 0.65 ESR2 (0.44) ESR2DRD2DRD3DRD4HRH3
SCHEMBL10930535 0.65 ESR2 (0.50) ESR2DRD2DRD3DRD4
SCHEMBL10932075 0.65 ESR2 (0.46) ESR2DRD2DRD3DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020120539-A1 NEW PYRROLIDINE-2-CARBOXYLIC ACID DERIVATIVES FOR TREATING PAIN AND PAIN RELATED CONDITIONS ESTEVE PHARMACEUTICALS, S.A. (ES) 2020-06-18 WO disclosed